Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS10009628HBVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS10031895HBVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS10038323HBVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS10041715HBVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS10041716HBVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS10043306HBVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS10052325HBVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS10043307HBVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS30078052HIVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS30085943HIVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TCGA Plot Options
Drug Information
GeneRARB
DrugBank IDDB12808
Drug NameTrifarotene
Target IDBE0000206
UniProt IDP10826
Regulation Typeagonist
PubMed IDs29974453
CitationsAubert J, Piwnica D, Bertino B, Blanchet-Rethore S, Carlavan I, Deret S, Dreno B, Gamboa B, Jomard A, Luzy AP, Mauvais P, Mounier C, Pascau J, Pelisson I, Portal T, Rivier M, Rossio P, Thoreau E, Vial E, Voegel JJ: Nonclinical and human pharmacology of the potent and selective topical retinoic acid receptor-gamma agonist trifarotene. Br J Dermatol. 2018 Aug;179(2):442-456. doi: 10.1111/bjd.16719. Epub 2018 Jul 4.
GroupsApproved; Investigational
Direct ClassificationM-terphenyls
SMILESCC(C)(C)C1=CC(=CC=C1N1CCCC1)C1=CC(=CC=C1OCCO)C1=CC=C(C=C1)C(O)=O
Pathways
PharmGKB
ChEMBLCHEMBL3707313