Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS30014534HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS30001571HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS30011269HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS30086715HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS30083245HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS30017988HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS30023982HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS30023983HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS30023984HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS30021093HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TCGA Plot Options
Drug Information
GenePDE4B
DrugBank IDDB05219
Drug NameCrisaborole
Target IDBE0000487
UniProt IDQ07343
Regulation Typeinhibitor
PubMed IDs22841723
CitationsFreund YR, Akama T, Alley MR, Antunes J, Dong C, Jarnagin K, Kimura R, Nieman JA, Maples KR, Plattner JJ, Rock F, Sharma R, Singh R, Sanders V, Zhou Y: Boron-based phosphodiesterase inhibitors show novel binding of boron to PDE4 bimetal center. FEBS Lett. 2012 Sep 21;586(19):3410-4. doi: 10.1016/j.febslet.2012.07.058. Epub 2012 Jul 25.
GroupsApproved; Investigational
Direct ClassificationDiarylethers
SMILESOB1OCC2=C1C=CC(OC1=CC=C(C=C1)C#N)=C2
Pathways
PharmGKB
ChEMBLCHEMBL484785