Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS30003501HIVENSG00000121807.7protein_codingCCR2NoNo729230P41597
TVIS30003502HIVENSG00000121807.7protein_codingCCR2NoNo729230P41597
TCGA Plot Options
Drug Information
GeneCCR2
DrugBank IDDB11758
Drug NameCenicriviroc
Target IDBE0003387
UniProt IDP41597
Regulation Typeinhibitor
PubMed IDs33849361
CitationsFiorucci S, Biagioli M, Baldoni M, Ricci P, Sepe V, Zampella A, Distrutti E: The identification of farnesoid X receptor modulators as treatment options for nonalcoholic fatty liver disease. Expert Opin Drug Discov. 2021 Oct;16(10):1193-1208. doi: 10.1080/17460441.2021.1916465. Epub 2021 May 5.
GroupsInvestigational
Direct ClassificationBenzazocines
SMILESCCCCOCCOC1=CC=C(C=C1)C1=CC2=C(C=C1)N(CC(C)C)CCCC(=C/2)C(=O)NC1=CC=C(C=C1)[S@@](=O)CC1=CN=CN1CCC
Pathways
PharmGKB
ChEMBLCHEMBL2110727