Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS20019921HPVENSG00000197561.7protein_codingELANENoNo1991P08246
TVIS20019922HPVENSG00000197561.7protein_codingELANENoNo1991P08246
TCGA Plot Options
Drug Information
GeneELANE
DrugBank IDDB03925
Drug NameFreselestat
Target IDBE0000394
UniProt IDP08246
Regulation Typeinhibitor
PubMed IDs11752352; 14530017
CitationsChen X, Ji ZL, Chen YZ: TTD: Therapeutic Target Database. Nucleic Acids Res. 2002 Jan 1;30(1):412-5.@@Yoshimura Y, Hiramatsu Y, Sato Y, Homma S, Enomoto Y, Jikuya T, Sakakibara Y: ONO-6818, a novel, potent neutrophil elastase inhibitor, reduces inflammatory mediators during simulated extracorporeal circulation. Ann Thorac Surg. 2003 Oct;76(4):1234-9.
GroupsExperimental; Investigational
Direct ClassificationPyrimidones
SMILESCC(C)[C@@H](NC(=O)CN1C(=O)C(N)=CN=C1C1=CC=CC=C1)[C@@H](O)C1=NN=C(O1)C(C)(C)C
Pathways
PharmGKB
ChEMBL