Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS30056468HIVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS30056469HIVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS30056470HIVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS30056471HIVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS20001736HPVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS20018964HPVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS20056614HPVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS20056970HPVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS20057260HPVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TVIS20056508HPVENSG00000077092.20protein_codingRARBNoNo5915P10826
Q5QHG3
Q86UC5
TCGA Plot Options
Drug Information
GeneRARB
DrugBank IDDB12808
Drug NameTrifarotene
Target IDBE0000206
UniProt IDP10826
Regulation Typeagonist
PubMed IDs29974453
CitationsAubert J, Piwnica D, Bertino B, Blanchet-Rethore S, Carlavan I, Deret S, Dreno B, Gamboa B, Jomard A, Luzy AP, Mauvais P, Mounier C, Pascau J, Pelisson I, Portal T, Rivier M, Rossio P, Thoreau E, Vial E, Voegel JJ: Nonclinical and human pharmacology of the potent and selective topical retinoic acid receptor-gamma agonist trifarotene. Br J Dermatol. 2018 Aug;179(2):442-456. doi: 10.1111/bjd.16719. Epub 2018 Jul 4.
GroupsApproved; Investigational
Direct ClassificationM-terphenyls
SMILESCC(C)(C)C1=CC(=CC=C1N1CCCC1)C1=CC(=CC=C1OCCO)C1=CC=C(C=C1)C(O)=O
Pathways
PharmGKB
ChEMBLCHEMBL3707313