Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS30011232HIVENSG00000116478.13protein_codingHDAC1YesNo3065Q13547
Q6IT96
TVIS30011233HIVENSG00000116478.13protein_codingHDAC1YesNo3065Q13547
Q6IT96
TVIS30023050HIVENSG00000116478.13protein_codingHDAC1YesNo3065Q13547
Q6IT96
TVIS30023051HIVENSG00000116478.13protein_codingHDAC1YesNo3065Q13547
Q6IT96
TVIS30023052HIVENSG00000116478.13protein_codingHDAC1YesNo3065Q13547
Q6IT96
TVIS30023053HIVENSG00000116478.13protein_codingHDAC1YesNo3065Q13547
Q6IT96
TVIS30023054HIVENSG00000116478.13protein_codingHDAC1YesNo3065Q13547
Q6IT96
TVIS30023055HIVENSG00000116478.13protein_codingHDAC1YesNo3065Q13547
Q6IT96
TVIS30023056HIVENSG00000116478.13protein_codingHDAC1YesNo3065Q13547
Q6IT96
TVIS30023057HIVENSG00000116478.13protein_codingHDAC1YesNo3065Q13547
Q6IT96
TCGA Plot Options
Drug Information
GeneHDAC1
DrugBank IDDB11830
Drug NameMocetinostat
Target IDBE0002365
UniProt IDQ13547
Regulation Type
PubMed IDs17455259; 17868033
CitationsBeckers T, Burkhardt C, Wieland H, Gimmnich P, Ciossek T, Maier T, Sanders K: Distinct pharmacological properties of second generation HDAC inhibitors with the benzamide or hydroxamate head group. Int J Cancer. 2007 Sep 1;121(5):1138-48.@@Khan N, Jeffers M, Kumar S, Hackett C, Boldog F, Khramtsov N, Qian X, Mills E, Berghs SC, Carey N, Finn PW, Collins LS, Tumber A, Ritchie JW, Jensen PB, Lichenstein HS, Sehested M: Determination of the class and isoform selectivity of small-molecule histone deacetylase inhibitors. Biochem J. 2008 Jan 15;409(2):581-9.
GroupsInvestigational
Direct ClassificationBenzanilides
SMILESNC1=CC=CC=C1NC(=O)C1=CC=C(CNC2=NC=CC(=N2)C2=CC=CN=C2)C=C1
Pathways
PharmGKB
ChEMBLCHEMBL272980