Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS30023985HIVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS20007444HPVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS20036920HPVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS20039414HPVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS20022219HPVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS20022256HPVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS20022231HPVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS20022242HPVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS20022221HPVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TVIS20022222HPVENSG00000184588.18protein_codingPDE4BNoNo5142Q07343
X5DNX5
X5DR82
TCGA Plot Options
Drug Information
GenePDE4B
DrugBank IDDB05219
Drug NameCrisaborole
Target IDBE0000487
UniProt IDQ07343
Regulation Typeinhibitor
PubMed IDs22841723
CitationsFreund YR, Akama T, Alley MR, Antunes J, Dong C, Jarnagin K, Kimura R, Nieman JA, Maples KR, Plattner JJ, Rock F, Sharma R, Singh R, Sanders V, Zhou Y: Boron-based phosphodiesterase inhibitors show novel binding of boron to PDE4 bimetal center. FEBS Lett. 2012 Sep 21;586(19):3410-4. doi: 10.1016/j.febslet.2012.07.058. Epub 2012 Jul 25.
GroupsApproved; Investigational
Direct ClassificationDiarylethers
SMILESOB1OCC2=C1C=CC(OC1=CC=C(C=C1)C#N)=C2
Pathways
PharmGKB
ChEMBLCHEMBL484785