Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS10020921HBVENSG00000101958.14protein_codingGLRA2NoNo2742P23416
TVIS10020920HBVENSG00000101958.14protein_codingGLRA2NoNo2742P23416
TVIS10014897HBVENSG00000101958.14protein_codingGLRA2NoNo2742P23416
TVIS10014898HBVENSG00000101958.14protein_codingGLRA2NoNo2742P23416
TVIS10020940HBVENSG00000101958.14protein_codingGLRA2NoNo2742P23416
TVIS10031645HBVENSG00000101958.14protein_codingGLRA2NoNo2742P23416
TVIS10031646HBVENSG00000101958.14protein_codingGLRA2NoNo2742P23416
TVIS10033377HBVENSG00000101958.14protein_codingGLRA2NoNo2742P23416
TVIS10042368HBVENSG00000101958.14protein_codingGLRA2NoNo2742P23416
TVIS30072819HIVENSG00000101958.14protein_codingGLRA2NoNo2742P23416
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Drug Information
GeneGLRA2
DrugBank IDDB00466
Drug NamePicrotoxin
Target IDBE0000745
UniProt IDP23416
Regulation Typeantagonist
PubMed IDs17714449; 17405877
CitationsYang Z, Cromer BA, Harvey RJ, Parker MW, Lynch JW: A proposed structural basis for picrotoxinin and picrotin binding in the glycine receptor pore. J Neurochem. 2007 Oct;103(2):580-9. Epub 2007 Aug 20.@@Wang DS, Buckinx R, Lecorronc H, Mangin JM, Rigo JM, Legendre P: Mechanisms for picrotoxinin and picrotin blocks of alpha2 homomeric glycine receptors. J Biol Chem. 2007 Jun 1;282(22):16016-35. Epub 2007 Apr 3.
GroupsExperimental
Direct ClassificationFuropyrans
SMILES[H][C@@]12OC(=O)[C@@]34OC3C[C@@](O)(C3[C@@H](C1OC3=O)C(C)=C)[C@@]24C.[H][C@@]12C[C@@]3(O)C4[C@@H](C(OC4=O)[C@@]4([H])OC(=O)[C@]1(O2)[C@@]34C)C(C)(C)O
Pathways
PharmGKBPA164777007
ChEMBLCHEMBL1908342