Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS46000368BKPyvENSG00000138823.14protein_codingMTTPNoNo4547E9PBP6
P55157
TVIS30060587HIVENSG00000138823.14protein_codingMTTPNoNo4547E9PBP6
P55157
TVIS20058865HPVENSG00000138823.14protein_codingMTTPNoNo4547E9PBP6
P55157
TCGA Plot Options
Drug Information
GeneMTTP
DrugBank IDDB05678
Drug NameSLx-4090
Target IDBE0000232
UniProt IDP55157
Regulation Typeinhibitor
PubMed IDs21406547
CitationsKim E, Campbell S, Schueller O, Wong E, Cole B, Kuo J, Ellis J, Ferkany J, Sweetnam P: A small-molecule inhibitor of enterocytic microsomal triglyceride transfer protein, SLx-4090: biochemical, pharmacodynamic, pharmacokinetic, and safety profile. J Pharmacol Exp Ther. 2011 Jun;337(3):775-85. doi: 10.1124/jpet.110.177527. Epub 2011 Mar 15.
GroupsInvestigational
Direct Classification
SMILESCOC1=CC=CC(C(=O)NC2=CC3=C(CN(CC3)C(=O)OC3=CC=CC=C3)C=C2)=C1C1=CC=C(C=C1)C(F)(F)F
Pathways
PharmGKB
ChEMBL