Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS10011228HBVENSG00000171608.18protein_codingPIK3CDYesNo5293O00329
TVIS30005072HIVENSG00000171608.18protein_codingPIK3CDYesNo5293O00329
TVIS30005073HIVENSG00000171608.18protein_codingPIK3CDYesNo5293O00329
TVIS30001457HIVENSG00000171608.18protein_codingPIK3CDYesNo5293O00329
TVIS30011160HIVENSG00000171608.18protein_codingPIK3CDYesNo5293O00329
TVIS30014456HIVENSG00000171608.18protein_codingPIK3CDYesNo5293O00329
TVIS30011161HIVENSG00000171608.18protein_codingPIK3CDYesNo5293O00329
TVIS30005074HIVENSG00000171608.18protein_codingPIK3CDYesNo5293O00329
TVIS30001458HIVENSG00000171608.18protein_codingPIK3CDYesNo5293O00329
TVIS30011162HIVENSG00000171608.18protein_codingPIK3CDYesNo5293O00329
TCGA Plot Options
Drug Information
GenePIK3CD
DrugBank IDDB05552
Drug NameTG100-115
Target IDBE0002406
UniProt IDO00329
Regulation Typeinhibitor
PubMed IDs17685602
CitationsPalanki MS, Dneprovskaia E, Doukas J, Fine RM, Hood J, Kang X, Lohse D, Martin M, Noronha G, Soll RM, Wrasidlo W, Yee S, Zhu H: Discovery of 3,3'-(2,4-diaminopteridine-6,7-diyl)diphenol as an isozyme-selective inhibitor of PI3K for the treatment of ischemia reperfusion injury associated with myocardial infarction. J Med Chem. 2007 Sep 6;50(18):4279-94. doi: 10.1021/jm051056c. Epub 2007 Aug 9.
GroupsInvestigational
Direct Classification
SMILESNC1=NC(N)=C2N=C(C3=CC=CC(O)=C3)C(=NC2=N1)C1=CC(O)=CC=C1
Pathways
PharmGKB
ChEMBLCHEMBL230011