Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS30087724HIVENSG00000108878.5protein_codingCACNG1NoNo786Q06432
TVIS30044813HIVENSG00000108878.5protein_codingCACNG1NoNo786Q06432
TVIS20036507HPVENSG00000108878.5protein_codingCACNG1NoNo786Q06432
TVIS44023880HTLV-1ENSG00000108878.5protein_codingCACNG1NoNo786Q06432
TCGA Plot Options
Drug Information
GeneCACNG1
DrugBank IDDB00528
Drug NameLercanidipine
Target IDBE0000679
UniProt IDQ06432
Regulation Typeinhibitor
PubMed IDs17139284; 17016423; 19619074
CitationsOverington JP, Al-Lazikani B, Hopkins AL: How many drug targets are there? Nat Rev Drug Discov. 2006 Dec;5(12):993-6.@@Imming P, Sinning C, Meyer A: Drugs, their targets and the nature and number of drug targets. Nat Rev Drug Discov. 2006 Oct;5(10):821-34.@@Burnier M, Pruijm M, Wuerzner G: Treatment of essential hypertension with calcium channel blockers: what is the place of lercanidipine? Expert Opin Drug Metab Toxicol. 2009 Aug;5(8):981-7. doi: 10.1517/17425250903085135.
GroupsApproved; Investigational
Direct ClassificationDiphenylmethanes
SMILESCOC(=O)C1=C(C)NC(C)=C(C1C1=CC(=CC=C1)[N+]([O-])=O)C(=O)OC(C)(C)CN(C)CCC(C1=CC=CC=C1)C1=CC=CC=C1
Pathways
PharmGKBPA164769058
ChEMBLCHEMBL250270