Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS30013507HIVENSG00000164850.16protein_codingGPER1NoNo2852Q99527
TVIS20007078HPVENSG00000164850.16protein_codingGPER1NoNo2852Q99527
TCGA Plot Options
Drug Information
GeneGPER1
DrugBank IDDB13953
Drug NameEstradiol benzoate
Target IDBE0003446
UniProt IDQ99527
Regulation Type
PubMed IDs17088055
CitationsThomas P, Dong J: Binding and activation of the seven-transmembrane estrogen receptor GPR30 by environmental estrogens: a potential novel mechanism of endocrine disruption. J Steroid Biochem Mol Biol. 2006 Dec;102(1-5):175-9. Epub 2006 Nov 7.
GroupsApproved; Investigational; Vet_approved
Direct ClassificationEstrane steroids
SMILES[H][C@]1(O)CC[C@@]2([H])[C@]3([H])CCC4=CC(OC(=O)C5=CC=CC=C5)=CC=C4[C@@]3([H])CC[C@]12C
Pathways
PharmGKB
ChEMBLCHEMBL282575