Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS10019549HBVENSG00000182578.14protein_codingCSF1RNoNo1436P07333
TVIS10036143HBVENSG00000182578.14protein_codingCSF1RNoNo1436P07333
TVIS10062766HBVENSG00000182578.14protein_codingCSF1RNoNo1436P07333
TCGA Plot Options
Drug Information
GeneCSF1R
DrugBank IDDB12978
Drug NamePexidartinib
Target IDBE0000853
UniProt IDP07333
Regulation Typeinhibitor
PubMed IDs28716061
CitationsCannarile MA, Weisser M, Jacob W, Jegg AM, Ries CH, Ruttinger D: Colony-stimulating factor 1 receptor (CSF1R) inhibitors in cancer therapy. J Immunother Cancer. 2017 Jul 18;5(1):53. doi: 10.1186/s40425-017-0257-y.
GroupsApproved; Investigational
Direct ClassificationPyrrolopyridines
SMILESFC(F)(F)C1=CC=C(CNC2=NC=C(CC3=CNC4=NC=C(Cl)C=C34)C=C2)C=N1
Pathways
PharmGKB
ChEMBLCHEMBL3813873