Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS30049098HIVENSG00000087088.21protein_codingBAXNoNo581I6LPK7
Q07812
Q5ZPJ0
Q5ZPJ1
TVIS44051578HTLV-1ENSG00000087088.21protein_codingBAXNoNo581I6LPK7
Q07812
Q5ZPJ0
Q5ZPJ1
TCGA Plot Options
Drug Information
GeneBAX
DrugBank IDDB12756
Drug NameTAK-901
Target IDBE0010137
UniProt IDQ07812
Regulation Typeactivator
PubMed IDs28179288
CitationsMurai S, Matuszkiewicz J, Okuzono Y, Miya H, DE Jong R: Aurora B Inhibitor TAK-901 Synergizes with BCL-xL Inhibition by Inducing Active BAX in Cancer Cells. Anticancer Res. 2017 Feb;37(2):437-444. doi: 10.21873/anticanres.11335.
GroupsInvestigational
Direct ClassificationAlpha carbolines
SMILESCCS(=O)(=O)C1=CC=CC(=C1)C1=CC(C(=O)NC2CCN(C)CC2)=C(C)C2=C1C1=C(N2)N=CC(C)=C1
Pathways
PharmGKB
ChEMBLCHEMBL3544932