Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS10002892HBVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS10022331HBVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS10029333HBVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS10045058HBVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20005969HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20008720HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20041792HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20022109HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20022108HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20056982HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TCGA Plot Options
Drug Information
GeneHTR1F
DrugBank IDDB00216
Drug NameEletriptan
Target IDBE0000460
UniProt IDP30939
Regulation Typeagonist
PubMed IDs10193663; 11834243; 15185063
CitationsNapier C, Stewart M, Melrose H, Hopkins B, McHarg A, Wallis R: Characterisation of the 5-HT receptor binding profile of eletriptan and kinetics of [3H]eletriptan binding at human 5-HT1B and 5-HT1D receptors. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.@@Bhalla P, Sharma HS, Wurch T, Pauwels PJ, Saxena PR: Molecular cloning and expression of the porcine trigeminal ganglion cDNA encoding a 5-ht(1F) receptor. Eur J Pharmacol. 2002 Feb 1;436(1-2):23-33.@@Jahnichen S, Radtke OA, Pertz HH: Involvement of 5-HT1B receptors in triptan-induced contractile responses in guinea-pig isolated iliac artery. Naunyn Schmiedebergs Arch Pharmacol. 2004 Jul;370(1):54-63. Epub 2004 Jun 8.
GroupsApproved; Investigational
Direct Classification3-alkylindoles
SMILESCN1CCC[C@@H]1CC1=CNC2=C1C=C(CCS(=O)(=O)C1=CC=CC=C1)C=C2
Pathways
PharmGKBPA134687947
ChEMBLCHEMBL1510