Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS30060134HIVENSG00000109163.7protein_codingGNRHRNoNo2798P30968
TVIS30060135HIVENSG00000109163.7protein_codingGNRHRNoNo2798P30968
TVIS20009946HPVENSG00000109163.7protein_codingGNRHRNoNo2798P30968
TCGA Plot Options
Drug Information
GeneGNRHR
DrugBank IDDB11853
Drug NameRelugolix
Target IDBE0000203
UniProt IDP30968
Regulation Typeantagonist
PubMed IDs
Citations
GroupsApproved; Investigational
Direct ClassificationN-phenylureas
SMILESCONC(=O)NC1=CC=C(C=C1)C1=C(CN(C)C)C2=C(S1)N(CC1=C(F)C=CC=C1F)C(=O)N(C2=O)C1=CC=C(OC)N=N1
Pathways
PharmGKB
ChEMBLCHEMBL1800159