Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS30060134HIVENSG00000109163.7protein_codingGNRHRNoNo2798P30968
TVIS30060135HIVENSG00000109163.7protein_codingGNRHRNoNo2798P30968
TVIS20009946HPVENSG00000109163.7protein_codingGNRHRNoNo2798P30968
TCGA Plot Options
Drug Information
GeneGNRHR
DrugBank IDDB17083
Drug NameLinzagolix
Target IDBE0000203
UniProt IDP30968
Regulation Typeantagonist
PubMed IDs35690889
CitationsTezuka M, Tamai Y, Kuramochi Y, Kobayashi K, Fushimi N, Kiguchi S: Pharmacological characterization of linzagolix, a novel, orally active, non-peptide antagonist of gonadotropin-releasing hormone receptors. Clin Exp Pharmacol Physiol. 2022 Oct;49(10):1082-1093. doi: 10.1111/1440-1681.13688. Epub 2022 Jul 12.
GroupsApproved
Direct Classification
SMILESCOC1=C(COC2=C(OC)C=C(F)C(=C2)N2C(=O)NC3=CSC(C(O)=O)=C3C2=O)C(F)=C(F)C=C1
Pathways
PharmGKB
ChEMBLCHEMBL3668014