Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS20034457HPVENSG00000132170.24protein_codingPPARGYesNo5468D2KUA6
E9PFX5
P37231
Q4W448
TVIS44022053HTLV-1ENSG00000132170.24protein_codingPPARGYesNo5468D2KUA6
E9PFX5
P37231
Q4W448
TVIS44006310HTLV-1ENSG00000132170.24protein_codingPPARGYesNo5468D2KUA6
E9PFX5
P37231
Q4W448
TVIS44022055HTLV-1ENSG00000132170.24protein_codingPPARGYesNo5468D2KUA6
E9PFX5
P37231
Q4W448
TCGA Plot Options
Drug Information
GenePPARG
DrugBank IDDB06521
Drug NameErtiprotafib
Target IDBE0000215
UniProt IDP37231
Regulation Type
PubMed IDs15475571
CitationsErbe DV, Wang S, Zhang YL, Harding K, Kung L, Tam M, Stolz L, Xing Y, Furey S, Qadri A, Klaman LD, Tobin JF: Ertiprotafib improves glycemic control and lowers lipids via multiple mechanisms. Mol Pharmacol. 2005 Jan;67(1):69-77. Epub 2004 Oct 8.
GroupsInvestigational
Direct ClassificationNaphthothiophenes
SMILESCC1=C(C)C2=C(C3=CC(C)=C(O[C@H](CC4=CC=CC=C4)C(O)=O)C(C)=C3)C3=CC=CC=C3C(Br)=C2S1
Pathways
PharmGKB
ChEMBLCHEMBL184041