Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS10036751HBVENSG00000136160.17protein_codingEDNRBNoNo1910P24530
TVIS10050050HBVENSG00000136160.17protein_codingEDNRBNoNo1910P24530
TVIS30035474HIVENSG00000136160.17protein_codingEDNRBNoNo1910P24530
TVIS20046672HPVENSG00000136160.17protein_codingEDNRBNoNo1910P24530
TCGA Plot Options
Drug Information
GeneEDNRB
DrugBank IDDB06558
Drug NameTezosentan
Target IDBE0000043
UniProt IDP24530
Regulation Type
PubMed IDs15542526
CitationsUrbanowicz W, Sogni P, Moreau R, Tazi KA, Barriere E, Poirel O, Martin A, Guimont MC, Cazals-Hatem D, Lebrec D: Tezosentan, an endothelin receptor antagonist, limits liver injury in endotoxin challenged cirrhotic rats. Gut. 2004 Dec;53(12):1844-9.
GroupsInvestigational
Direct ClassificationPyridinylpyrimidines
SMILESCOC1=CC=CC=C1OC1=C(NS(=O)(=O)C2=NC=C(C=C2)C(C)C)N=C(N=C1OCCO)C1=CC(=NC=C1)C1=NNN=N1
Pathways
PharmGKB
ChEMBLCHEMBL61780