Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS42001512EBVENSG00000112038.18protein_codingOPRM1NoNo4988B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
TVIS10012006HBVENSG00000112038.18protein_codingOPRM1NoNo4988B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
TVIS10007858HBVENSG00000112038.18protein_codingOPRM1NoNo4988B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
TVIS10008487HBVENSG00000112038.18protein_codingOPRM1NoNo4988B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
TVIS10009685HBVENSG00000112038.18protein_codingOPRM1NoNo4988B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
TVIS10010472HBVENSG00000112038.18protein_codingOPRM1NoNo4988B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
TVIS10010870HBVENSG00000112038.18protein_codingOPRM1NoNo4988B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
TVIS10011363HBVENSG00000112038.18protein_codingOPRM1NoNo4988B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
TVIS10011435HBVENSG00000112038.18protein_codingOPRM1NoNo4988B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
TVIS10013160HBVENSG00000112038.18protein_codingOPRM1NoNo4988B8K2Q5
G8XRH4
G8XRH5
L0E130
P35372
TCGA Plot Options
Drug Information
GeneOPRM1
DrugBank IDDB14146
Drug NameLoxicodegol
Target IDBE0000770
UniProt IDP35372
Regulation Typeagonist
PubMed IDs28778859
CitationsMiyazaki T, Choi IY, Rubas W, Anand NK, Ali C, Evans J, Gursahani H, Hennessy M, Kim G, McWeeney D, Pfeiffer J, Quach P, Gauvin D, Riley TA, Riggs JA, Gogas K, Zalevsky J, Doberstein SK: NKTR-181: A Novel Mu-Opioid Analgesic with Inherently Low Abuse Potential. J Pharmacol Exp Ther. 2017 Oct;363(1):104-113. doi: 10.1124/jpet.117.243030. Epub 2017 Aug 4.
GroupsInvestigational
Direct Classification
SMILES[H][C@@]12OC3=C(OC)C=CC4=C3[C@@]11CCN(C)[C@]([H])(C4)[C@]1(O)CC[C@]2([H])OCCOCCOCCOCCOCCOCCOC
Pathways
PharmGKB
ChEMBL