Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS10019723HBVENSG00000091831.25protein_codingESR1YesNo2099A0A125SXW3
G4XH65
H0Y4W6
P03372
TVIS10020557HBVENSG00000091831.25protein_codingESR1YesNo2099A0A125SXW3
G4XH65
H0Y4W6
P03372
TVIS10048572HBVENSG00000091831.25protein_codingESR1YesNo2099A0A125SXW3
G4XH65
H0Y4W6
P03372
TVIS30009202HIVENSG00000091831.25protein_codingESR1YesNo2099A0A125SXW3
G4XH65
H0Y4W6
P03372
TVIS30087612HIVENSG00000091831.25protein_codingESR1YesNo2099A0A125SXW3
G4XH65
H0Y4W6
P03372
TVIS30066142HIVENSG00000091831.25protein_codingESR1YesNo2099A0A125SXW3
G4XH65
H0Y4W6
P03372
TVIS30066143HIVENSG00000091831.25protein_codingESR1YesNo2099A0A125SXW3
G4XH65
H0Y4W6
P03372
TVIS30066144HIVENSG00000091831.25protein_codingESR1YesNo2099A0A125SXW3
G4XH65
H0Y4W6
P03372
TVIS20006531HPVENSG00000091831.25protein_codingESR1YesNo2099A0A125SXW3
G4XH65
H0Y4W6
P03372
TVIS20060785HPVENSG00000091831.25protein_codingESR1YesNo2099A0A125SXW3
G4XH65
H0Y4W6
P03372
TCGA Plot Options
Drug Information
GeneESR1
DrugBank IDDB09070
Drug NameTibolone
Target IDBE0000123
UniProt IDP03372
Regulation Typeantagonist
PubMed IDs19464167
CitationsEscande A, Servant N, Rabenoelina F, Auzou G, Kloosterboer H, Cavailles V, Balaguer P, Maudelonde T: Regulation of activities of steroid hormone receptors by tibolone and its primary metabolites. J Steroid Biochem Mol Biol. 2009 Aug;116(1-2):8-14. doi: 10.1016/j.jsbmb.2009.03.008. Epub 2009 Apr 2.
GroupsApproved; Investigational
Direct ClassificationOxosteroids
SMILES[H][C@@]12CC[C@@](O)(C#C)[C@@]1(C)CC[C@]1([H])C3=C(CC(=O)CC3)C[C@@]([H])(C)[C@@]21[H]
Pathways
PharmGKB
ChEMBLCHEMBL2103774