Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS10037354HBVENSG00000080644.16protein_codingCHRNA3NoNo1136P32297
TVIS10032120HBVENSG00000080644.16protein_codingCHRNA3NoNo1136P32297
TVIS10039140HBVENSG00000080644.16protein_codingCHRNA3NoNo1136P32297
TVIS30039129HIVENSG00000080644.16protein_codingCHRNA3NoNo1136P32297
TCGA Plot Options
Drug Information
GeneCHRNA3
DrugBank IDDB01273
Drug NameVarenicline
Target IDBE0003585
UniProt IDP32297
Regulation Typepartial agonist
PubMed IDs16766716
CitationsMihalak KB, Carroll FI, Luetje CW: Varenicline is a partial agonist at alpha4beta2 and a full agonist at alpha7 neuronal nicotinic receptors. Mol Pharmacol. 2006 Sep;70(3):801-5. Epub 2006 Jun 9.
GroupsApproved; Investigational
Direct Classification
SMILESC1C2CNCC1C1=C2C=C2N=CC=NC2=C1
Pathways
PharmGKBPA164781343
ChEMBLCHEMBL1396