Target Gene Table
VIS IDVirusEnsembl IDGene TypeTarget GeneOncogeneTumor Suppressor GeneNCBI IDUniprot ID
TVIS10002892HBVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS10022331HBVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS10029333HBVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS10045058HBVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20005969HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20008720HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20041792HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20022109HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20022108HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TVIS20056982HPVENSG00000179097.7protein_codingHTR1FNoNo3355P30939
TCGA Plot Options
Drug Information
GeneHTR1F
DrugBank IDDB00952
Drug NameNaratriptan
Target IDBE0000460
UniProt IDP30939
Regulation Typeagonist
PubMed IDs11752352; 14725972; 11152011; 12463278; 15320857; 14614913; 12434581
CitationsChen X, Ji ZL, Chen YZ: TTD: Therapeutic Target Database. Nucleic Acids Res. 2002 Jan 1;30(1):412-5.@@Hoskin KL, Lambert GA, Donaldson C, Zagami AS: The 5-hydroxytryptamine1B/1D/1F receptor agonists eletriptan and naratriptan inhibit trigeminovascular input to the nucleus tractus solitarius in the cat. Brain Res. 2004 Feb 13;998(1):91-9.@@Tfelt-Hansen P, De Vries P, Saxena PR: Triptans in migraine: a comparative review of pharmacology, pharmacokinetics and efficacy. Drugs. 2000 Dec;60(6):1259-87.@@Massiou H: Naratriptan. Curr Med Res Opin. 2001;17 Suppl 1:s51-3.@@Villalon CM, Centurion D, Valdivia LF, de Vries P, Saxena PR: Migraine: pathophysiology, pharmacology, treatment and future trends. Curr Vasc Pharmacol. 2003 Mar;1(1):71-84.@@Goadsby PJ, Classey JD: Evidence for serotonin (5-HT)1B, 5-HT1D and 5-HT1F receptor inhibitory effects on trigeminal neurons with craniovascular input. Neuroscience. 2003;122(2):491-8.@@Villalon CM, Centurion D, Valdivia LF, De Vries P, Saxena PR: An introduction to migraine: from ancient treatment to functional pharmacology and antimigraine therapy. Proc West Pharmacol Soc. 2002;45:199-210.
GroupsApproved; Investigational
Direct Classification3-alkylindoles
SMILESCNS(=O)(=O)CCC1=CC2=C(NC=C2C2CCN(C)CC2)C=C1
Pathways
PharmGKBPA450597
ChEMBLCHEMBL1278