DegronMD: protein-targeted degradation, mutation and drug response to degrons
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BSML
CPH
CGC
Degron:
DRRERDYTNLP
Uniprot ID:
P07333
Source protein:
Macrophage colony-stimulating factor 1 receptor
Source gene:
CSF1R
Class:
CBL_PTK
Location:
917:927
E3 ligase:
CBL
DEGRON score:
0.9362
ASA_SCORE:
88.1455
COIL:
0.7113
CONS_SCORE:
0.4113
DSS_SCORE:
0.6735
HELIX:
0.2
FCONS_SCORE:
1.1146
RIG_SCORE:
0.6894
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.R921W
TCGA-BA-A6DL
HNSC
TCGA
DRRERDYTNLP
CBL_PTK
0.7523
p.R921W
DO52035
HNSC
ICGC
DRRERDYTNLP
CBL_PTK
0.7523
p.R921W
SIDM01613
Colorectal Carcinoma
GDSC
DRRERDYTNLP
CBL_PTK
0.7523
p.E920D
SIDM00762
Non-Small Cell Lung Carcinoma
GDSC
DRRERDYTNLP
CBL_PTK
0.5647
p.E920D
SIDM01878
Non-Cancerous
GDSC
DRRERDYTNLP
CBL_PTK
0.5647
p.E920D
SIDM01007
T-Lymphoblastic Leukemia
GDSC
DRRERDYTNLP
CBL_PTK
0.5647
p.E920D
SIDM00333
Endometrial Carcinoma
GDSC
DRRERDYTNLP
CBL_PTK
0.5647
p.E920D
SIDM00382
Glioblastoma
GDSC
DRRERDYTNLP
CBL_PTK
0.5647
p.E920D
SIDM00053
Pancreatic Carcinoma
GDSC
DRRERDYTNLP
CBL_PTK
0.5647
p.E920D
SIDM00228
Thyroid Gland Carcinoma
GDSC
DRRERDYTNLP
CBL_PTK
0.5647
p.S932R
DO229038
LICA
ICGC
DRRERDYTNLP
CBL_PTK
0.1944
p.Q911E
TCGA-K4-A3WS
BLCA
TCGA
DRRERDYTNLP
CBL_PTK
0.1667
p.Q911E
DO480
BLCA
ICGC
DRRERDYTNLP
CBL_PTK
0.1667
p.G936S
DO228581
GACA
ICGC
DRRERDYTNLP
CBL_PTK
0.0833
p.G936S
DO233693
GACA
ICGC
DRRERDYTNLP
CBL_PTK
0.0833
p.G936S
SIDM01608
Endometrial Carcinoma
GDSC
DRRERDYTNLP
CBL_PTK
0.0833
p.G936S
ACH-000990
Endometrial/Uterine Cancer
CCLE
DRRERDYTNLP
CBL_PTK
0.0833
p.S937R
TCGA-24-1426
OV
TCGA
DRRERDYTNLP
CBL_PTK
0.0556
p.S937R
DO30010
OV
ICGC
DRRERDYTNLP
CBL_PTK
0.0556
p.S937G
SIDM00780
Colorectal Carcinoma
GDSC
DRRERDYTNLP
CBL_PTK
0.0556
p.S937G
ACH-000967
Colon/Colorectal Cancer
CCLE
DRRERDYTNLP
CBL_PTK
0.0556
p.S937G
ACH-001199
Colon/Colorectal Cancer
CCLE
DRRERDYTNLP
CBL_PTK
0.0556
p.S937G
ACH-001518
Endometrial/Uterine Cancer
CCLE
DRRERDYTNLP
CBL_PTK
0.0556
Showing 1 to 23 of 23 entries
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Drug responses associated with CSF1R mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
SIDM01007
ALL|lymphoblastic_leukemia
p.E920D (Yes)
GDSC
Sunitinib
2.0565
SIDM01007
ALL|lymphoblastic_leukemia
p.E920D (Yes)
GDSC
GW-2580
122.3043
SIDM01007
ALL|lymphoblastic_leukemia
p.E920D (Yes)
GDSC
Pazopanib
9.0608
SIDM01007
ALL|lymphoblastic_leukemia
p.E920D (Yes)
GDSC
Linifanib
4.2428
SIDM01007
ALL|lymphoblastic_leukemia
p.S188P (No)
GDSC
Sunitinib
2.0565
SIDM01007
ALL|lymphoblastic_leukemia
p.S188P (No)
GDSC
GW-2580
122.3043
SIDM01007
ALL|lymphoblastic_leukemia
p.S188P (No)
GDSC
Pazopanib
9.0608
SIDM01007
ALL|lymphoblastic_leukemia
p.S188P (No)
GDSC
Linifanib
4.2428
SIDM00451
ALL|lymphoblastic_T_cell_leukaemia
p.V138I (No)
GDSC
Sunitinib
2.8236
SIDM00451
ALL|lymphoblastic_T_cell_leukaemia
p.V138I (No)
GDSC
GW-2580
192.1361
SIDM00451
ALL|lymphoblastic_T_cell_leukaemia
p.V138I (No)
GDSC
Pazopanib
27.7744
SIDM00451
ALL|lymphoblastic_T_cell_leukaemia
p.V138I (No)
GDSC
Linifanib
9.659
SIDM00989
BLCA|bladder
p.S937_S938insGS (Yes)
GDSC
GW-2580
131.6997
SIDM00989
BLCA|bladder
p.S937_S938insGS (Yes)
GDSC
Pazopanib
27.8581
SIDM00989
BLCA|bladder
p.S937_S938insGS (Yes)
GDSC
Linifanib
9.0538
SIDM00940
BRCA|breast
p.R106Q (No)
GDSC
GW-2580
440.0921
SIDM00940
BRCA|breast
p.R106Q (No)
GDSC
Pazopanib
20.2904
SIDM00940
BRCA|breast
p.R106Q (No)
GDSC
Linifanib
21.8688
SIDM00630
BRCA|breast
p.Q970* (No)
GDSC
GW-2580
150.6293
SIDM00630
BRCA|breast
p.Q970* (No)
GDSC
Pazopanib
12.1881
SIDM00630
BRCA|breast
p.Q970* (No)
GDSC
Linifanib
29.1021
SIDM00673
BRCA|breast
p.P510A (No)
GDSC
GW-2580
288.5063
SIDM00673
BRCA|breast
p.P510A (No)
GDSC
Pazopanib
19.2114
SIDM00673
BRCA|breast
p.P510A (No)
GDSC
Linifanib
11.3311
SIDM00781
COREAD|large_intestine
p.P402fs*3 (No)
GDSC
Sunitinib
64.3744
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All proteins holding degron of DRRERDYTNLP
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
P07333
Macrophage colony-stimulating factor 1 receptor
CBL_PTK
917:927
DRRERDYTNLP
CBL
0.9362
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