DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
ARRFLARLT
Uniprot ID:
O75628
Source protein:
GTP-binding protein REM 1
Source gene:
REM1
Class:
DEG_APCC_DBOX_1
Location:
268:276
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.7594
ASA_SCORE:
90.5556
COIL:
0.1488
CONS_SCORE:
0.4716
DSS_SCORE:
0.4909
HELIX:
0.8493
FCONS_SCORE:
1.2237
RIG_SCORE:
0.7979
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.R269C
DO233270
GACA
ICGC
ARRFLARLT
DEG_APCC_DBOX_1
0.8301
p.R269C
DO222599
MELA
ICGC
ARRFLARLT
DEG_APCC_DBOX_1
0.8301
p.R270C
DO229232
THCA
ICGC
ARRFLARLT
DEG_APCC_DBOX_1
0.719
p.R274C
SIDM02039
Colorectal Carcinoma
GDSC
ARRFLARLT
DEG_APCC_DBOX_1
0.719
p.R274C
SIDM00053
Pancreatic Carcinoma
GDSC
ARRFLARLT
DEG_APCC_DBOX_1
0.719
p.R274C
ACH-000563
Lung Cancer
CCLE
ARRFLARLT
DEG_APCC_DBOX_1
0.719
p.R274C
ACH-002164
Pancreatic Cancer
CCLE
ARRFLARLT
DEG_APCC_DBOX_1
0.719
p.R274C
MZ1-PC
pancreas
COSMIC
ARRFLARLT
DEG_APCC_DBOX_1
0.719
p.R274H
DO12070
GBM
ICGC
ARRFLARLT
DEG_APCC_DBOX_1
0.7133
p.R270H
SIDM00151
Ovarian Carcinoma
GDSC
ARRFLARLT
DEG_APCC_DBOX_1
0.7133
p.R270H
ACH-000966
Ovarian Cancer
CCLE
ARRFLARLT
DEG_APCC_DBOX_1
0.7133
p.T276R
DO223065
ESCA
ICGC
ARRFLARLT
DEG_APCC_DBOX_1
0.6765
p.A268T
DO227668
COCA
ICGC
ARRFLARLT
DEG_APCC_DBOX_1
0.6028
p.R267H
DO234195
ESAD
ICGC
ARRFLARLT
DEG_APCC_DBOX_1
0.3056
p.R267H
SIDM00373
Endometrial Carcinoma
GDSC
ARRFLARLT
DEG_APCC_DBOX_1
0.3056
p.R267H
SIDM00422
Hodgkin's Lymphoma
GDSC
ARRFLARLT
DEG_APCC_DBOX_1
0.3056
p.R267H
SIDM00380
Acute Myeloid Leukemia
GDSC
ARRFLARLT
DEG_APCC_DBOX_1
0.3056
p.A265T
DO229275
THCA
ICGC
ARRFLARLT
DEG_APCC_DBOX_1
0.25
p.A280T
DO229213
THCA
ICGC
ARRFLARLT
DEG_APCC_DBOX_1
0.2222
p.P261L
SIDM00951
T-Lymphoblastic Leukemia
GDSC
ARRFLARLT
DEG_APCC_DBOX_1
0.1389
p.P261L
ACH-000251
Lung Cancer
CCLE
ARRFLARLT
DEG_APCC_DBOX_1
0.1389
p.A284T
DO229245
THCA
ICGC
ARRFLARLT
DEG_APCC_DBOX_1
0.1111
Showing 1 to 22 of 22 entries
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Drug responses associated with REM1 mutations
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Cancer
Mutation (In Degron?)
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Drug
IC50
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All proteins holding degron of ARRFLARLT
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
O75628
GTP-binding protein REM 1
DEG_APCC_DBOX_1
268:276
ARRFLARLT
APC,CDC20,FZR1
0.7594
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