DegronMD: protein-targeted degradation, mutation and drug response to degrons
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BSML
CPH
CGC
Degron:
FGRVWYRIL
Uniprot ID:
Q9H251
Source protein:
Cadherin-23
Source gene:
CDH23
Class:
DEG_MDM2_SWIB_1
Location:
1134:1142
E3 ligase:
MDM2
DEGRON score:
0.6575
ASA_SCORE:
48.8556
COIL:
0.2459
CONS_SCORE:
0.3214
DSS_SCORE:
0.2155
HELIX:
0.0083
FCONS_SCORE:
0.7079
RIG_SCORE:
0.8661
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.R1141C
DO222762
COCA
ICGC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.8301
p.R1141H
DO233109
GACA
ICGC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.8244
p.A1134T
DO42033
UCEC
ICGC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.7139
p.D1135N
DO2401
BRCA
ICGC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.6932
p.T1132M
DO41572
UCEC
ICGC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.2778
p.T1132M
ACH-001517
Endometrial/Uterine Cancer
CCLE
FGRVWYRIL
DEG_MDM2_SWIB_1
0.2778
p.G1144C
SIDM00420
Bladder Carcinoma
GDSC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.2778
p.L1129M
DO43907
UCEC
ICGC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.1944
p.Q1128H
DO229025
LICA
ICGC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.1667
p.R1150Q
Hs939-T
skin
COSMIC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.1111
p.R1151Q
SIDM00663
Melanoma
GDSC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.0833
p.R1151Q
Hs939-T
skin
COSMIC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.0833
p.E1124K
NUGC-3
stomach
COSMIC
FGRVWYRIL
DEG_MDM2_SWIB_1
0.0556
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Drug responses associated with CDH23 mutations
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Mutation (In Degron?)
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All proteins holding degron of FGRVWYRIL
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
Q9H251
Cadherin-23
DEG_MDM2_SWIB_1
1134:1142
FGRVWYRIL
MDM2
0.6575
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