DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
GRSMLETIK
Uniprot ID:
O43424
Source protein:
Glutamate receptor ionotropic, delta-2
Source gene:
GRID2
Class:
DEG_APCC_DBOX_1
Location:
366:374
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.8028
ASA_SCORE:
49.8111
COIL:
0.1391
CONS_SCORE:
0.4649
DSS_SCORE:
0.4875
HELIX:
0.8503
FCONS_SCORE:
1.2064
RIG_SCORE:
0.7513
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.R367C
TCGA-AX-A1CE
UCEC
TCGA
GRSMLETIK
DEG_APCC_DBOX_1
0.8301
p.R367C
TCGA-FI-A2D5
UCEC
TCGA
GRSMLETIK
DEG_APCC_DBOX_1
0.8301
p.R367C
SIDM01311
Esophageal Carcinoma
GDSC
GRSMLETIK
DEG_APCC_DBOX_1
0.8301
p.R367H
TCGA-W3-A828
SKCM
TCGA
GRSMLETIK
DEG_APCC_DBOX_1
0.8244
p.R367H
DO233272
GACA
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.8244
p.R367H
DO51273
SKCM
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.8244
p.G367C
DO37523
SKCM
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.76
p.P369L
DO223082
ESCA
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.7582
p.L368P
NCI-H2172
lung
COSMIC
GRSMLETIK
DEG_APCC_DBOX_1
0.7582
p.G374R
DO26617
LUSC
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.7568
p.G374D
DO45229
LIRI
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.7198
p.S368F
TCGA-EE-A29D
SKCM
TCGA
GRSMLETIK
DEG_APCC_DBOX_1
0.6871
p.M369T
TCGA-NH-A6GB
COAD
TCGA
GRSMLETIK
DEG_APCC_DBOX_1
0.6312
p.M369T
DO50092
COAD
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.6312
p.K374N
TCGA-EI-6917
READ
TCGA
GRSMLETIK
DEG_APCC_DBOX_1
0.5806
p.G365C
TCGA-77-8138
LUSC
TCGA
GRSMLETIK
DEG_APCC_DBOX_1
0.3056
p.G365C
DO233079
GACA
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.3056
p.G365C
DO26510
LUSC
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.3056
p.K361E
ACH-001061
Colon/Colorectal Cancer
CCLE
GRSMLETIK
DEG_APCC_DBOX_1
0.3056
p.Q364H
TCGA-22-5474
LUSC
TCGA
GRSMLETIK
DEG_APCC_DBOX_1
0.2778
p.S376F
BHT-101
thyroid
COSMIC
GRSMLETIK
DEG_APCC_DBOX_1
0.2778
p.P362S
TCGA-A5-A0G1
UCEC
TCGA
GRSMLETIK
DEG_APCC_DBOX_1
0.2222
p.P362S
TCGA-BS-A0T9
UCEC
TCGA
GRSMLETIK
DEG_APCC_DBOX_1
0.2222
p.P362S
DO41026
UCEC
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.2222
p.P362S
DO42472
UCEC
ICGC
GRSMLETIK
DEG_APCC_DBOX_1
0.2222
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Drug responses associated with GRID2 mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of GRSMLETIK
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
O43424
Glutamate receptor ionotropic, delta-2
DEG_APCC_DBOX_1
366:374
GRSMLETIK
APC,CDC20,FZR1
0.8028
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