DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
IKENM
Uniprot ID:
Q58F21
Source protein:
Bromodomain testis-specific protein
Source gene:
BRDT
Class:
DEG_APCC_KENBOX_2
Location:
245:249
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.6263
ASA_SCORE:
97.32
COIL:
0.7754
CONS_SCORE:
0.3045
DSS_SCORE:
0.5084
HELIX:
0.108
FCONS_SCORE:
0.9691
RIG_SCORE:
0.7272
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.K246Q
TCGA-B5-A0JY
UCEC
TCGA
IKENM
DEG_APCC_KENBOX_2
0.6944
p.K246Q
TCGA-BK-A6W3
UCEC
TCGA
IKENM
DEG_APCC_KENBOX_2
0.6944
p.K246Q
DO50076
UCEC
ICGC
IKENM
DEG_APCC_KENBOX_2
0.6944
p.K246Q
DO43041
UCEC
ICGC
IKENM
DEG_APCC_KENBOX_2
0.6944
p.K246N
TCGA-F5-6814
READ
TCGA
IKENM
DEG_APCC_KENBOX_2
0.6918
p.K246N
DO36556
READ
ICGC
IKENM
DEG_APCC_KENBOX_2
0.6918
p.P244H
TCGA-BR-8078
STAD
TCGA
IKENM
DEG_APCC_KENBOX_2
0.3056
p.P244H
DO38288
STAD
ICGC
IKENM
DEG_APCC_KENBOX_2
0.3056
p.K251N
TCGA-77-7335
LUSC
TCGA
IKENM
DEG_APCC_KENBOX_2
0.2778
p.K251N
TCGA-E6-A1LX
UCEC
TCGA
IKENM
DEG_APCC_KENBOX_2
0.2778
p.K251N
DO26707
LUSC
ICGC
IKENM
DEG_APCC_KENBOX_2
0.2778
p.K251N
DO41020
UCEC
ICGC
IKENM
DEG_APCC_KENBOX_2
0.2778
p.K251N
ACH-000993
Endometrial/Uterine Cancer
CCLE
IKENM
DEG_APCC_KENBOX_2
0.2778
p.K238N
DO228483
BRCA
ICGC
IKENM
DEG_APCC_KENBOX_2
0.25
p.K238N
DO227999
COCA
ICGC
IKENM
DEG_APCC_KENBOX_2
0.25
p.K238N
DO229010
COCA
ICGC
IKENM
DEG_APCC_KENBOX_2
0.25
p.K238N
DO229013
COCA
ICGC
IKENM
DEG_APCC_KENBOX_2
0.25
p.K238N
DO229016
COCA
ICGC
IKENM
DEG_APCC_KENBOX_2
0.25
p.K238N
DO229003
COCA
ICGC
IKENM
DEG_APCC_KENBOX_2
0.25
p.K238N
DO229346
LAML
ICGC
IKENM
DEG_APCC_KENBOX_2
0.25
p.K238N
DO229047
LICA
ICGC
IKENM
DEG_APCC_KENBOX_2
0.25
p.K238N
DO230993
LUSC
ICGC
IKENM
DEG_APCC_KENBOX_2
0.25
p.H242Y
NCI-H1770
lung
COSMIC
IKENM
DEG_APCC_KENBOX_2
0.25
p.V253L
NCI-H2110
lung
COSMIC
IKENM
DEG_APCC_KENBOX_2
0.2222
p.L254V
DO228221
MALY
ICGC
IKENM
DEG_APCC_KENBOX_2
0.1944
Showing 1 to 25 of 32 entries
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Drug responses associated with BRDT mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
SIDM00463
ALL|lymphoblastic_T_cell_leukaemia
p.I393T (No)
GDSC
JQ1
0.7368
SIDM00463
ALL|lymphoblastic_T_cell_leukaemia
p.I393T (No)
GDSC
JQ1
6.9137
SIDM00403
ALL|lymphoblastic_T_cell_leukaemia
p.S762L (No)
GDSC
JQ1
1.0227
SIDM00403
ALL|lymphoblastic_T_cell_leukaemia
p.S762L (No)
GDSC
JQ1
2.5702
SIDM00420
BLCA|bladder
p.S196L (No)
GDSC
JQ1
0.0632
SIDM00420
BLCA|bladder
p.S196L (No)
GDSC
JQ1
9.968
SIDM01042
BRCA|breast
p.D114G (No)
GDSC
JQ1
0.6062
SIDM01042
BRCA|breast
p.D114G (No)
GDSC
JQ1
8.8946
SIDM01042
BRCA|breast
p.D114G (No)
GDSC
JQ1
0.3458
SIDM00963
BRCA|breast
p.D414N (No)
GDSC
JQ1
2.135
SIDM00963
BRCA|breast
p.D414N (No)
GDSC
JQ1
25.7491
SIDM00963
BRCA|breast
p.D414N (No)
GDSC
JQ1
42.196
SIDM00194
COREAD|large_intestine
p.E685G (No)
GDSC
JQ1
10.9153
SIDM00150
COREAD|large_intestine
p.L437F (No)
GDSC
JQ1
0.6889
SIDM00150
COREAD|large_intestine
p.L437F (No)
GDSC
JQ1
14.8593
SIDM00534
COREAD|large_intestine
p.N470S (No)
GDSC
JQ1
2.062
SIDM00534
COREAD|large_intestine
p.N470S (No)
GDSC
JQ1
12.3123
SIDM00537
COREAD|large_intestine
p.R82H (No)
GDSC
JQ1
0.3119
SIDM00537
COREAD|large_intestine
p.R82H (No)
GDSC
JQ1
8.9937
SIDM00193
COREAD|large_intestine
p.S572L (No)
GDSC
JQ1
21.8249
SIDM00118
COREAD|large_intestine
p.K286N (No)
GDSC
JQ1
0.9581
SIDM00118
COREAD|large_intestine
p.K286N (No)
GDSC
JQ1
9.4882
SIDM00118
COREAD|large_intestine
p.E566* (No)
GDSC
JQ1
0.9581
SIDM00118
COREAD|large_intestine
p.E566* (No)
GDSC
JQ1
9.4882
SIDM00349
ESCA|oesophagus
p.S407C (No)
GDSC
JQ1
0.3163
Showing 1 to 25 of 86 entries
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All proteins holding degron of IKENM
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
Q58F21
Bromodomain testis-specific protein
DEG_APCC_KENBOX_2
245:249
IKENM
APC,CDC20,FZR1
0.6263
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