DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
LRRKLEELT
Uniprot ID:
Q9BV36
Source protein:
Melanophilin
Source gene:
MLPH
Class:
DEG_APCC_DBOX_1
Location:
385:393
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.9665
ASA_SCORE:
101.6333
COIL:
0.1633
CONS_SCORE:
0.6801
DSS_SCORE:
0.5702
HELIX:
0.8364
FCONS_SCORE:
1.2293
RIG_SCORE:
0.7537
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.N388T
DO13024
GBM
ICGC
LRRKLEELT
DEG_APCC_DBOX_1
0.7055
p.S397G
TCGA-EE-A2GN
SKCM
TCGA
LRRKLEELT
DEG_APCC_DBOX_1
0.6667
p.S397G
DO37896
SKCM
ICGC
LRRKLEELT
DEG_APCC_DBOX_1
0.6667
p.E391V
SIDM00656
Burkitt's Lymphoma
GDSC
LRRKLEELT
DEG_APCC_DBOX_1
0.6582
p.E391V
SIDM01318
Hepatocellular Carcinoma
GDSC
LRRKLEELT
DEG_APCC_DBOX_1
0.6582
p.E391V
SIDM00641
Burkitt's Lymphoma
GDSC
LRRKLEELT
DEG_APCC_DBOX_1
0.6582
p.E391V
SIDM01677
Non-Small Cell Lung Carcinoma
GDSC
LRRKLEELT
DEG_APCC_DBOX_1
0.6582
p.E391V
NAMALWA
haematopoietic_and_lymphoid_tissue
COSMIC
LRRKLEELT
DEG_APCC_DBOX_1
0.6582
p.E391K
TCGA-EA-A97N
CESC
TCGA
LRRKLEELT
DEG_APCC_DBOX_1
0.591
p.E391K
DO49935
CESC
ICGC
LRRKLEELT
DEG_APCC_DBOX_1
0.591
p.E391K
SIDM00656
Burkitt's Lymphoma
GDSC
LRRKLEELT
DEG_APCC_DBOX_1
0.591
p.E391K
SIDM01318
Hepatocellular Carcinoma
GDSC
LRRKLEELT
DEG_APCC_DBOX_1
0.591
p.E391K
SIDM00641
Burkitt's Lymphoma
GDSC
LRRKLEELT
DEG_APCC_DBOX_1
0.591
p.E391K
SIDM01677
Non-Small Cell Lung Carcinoma
GDSC
LRRKLEELT
DEG_APCC_DBOX_1
0.591
p.E391K
NAMALWA
haematopoietic_and_lymphoid_tissue
COSMIC
LRRKLEELT
DEG_APCC_DBOX_1
0.591
p.E390D
TCGA-B5-A3FC
UCEC
TCGA
LRRKLEELT
DEG_APCC_DBOX_1
0.5647
p.E390D
DO41871
UCEC
ICGC
LRRKLEELT
DEG_APCC_DBOX_1
0.5647
p.E383K
TCGA-VS-A958
CESC
TCGA
LRRKLEELT
DEG_APCC_DBOX_1
0.2778
p.E383K
DO51639
CESC
ICGC
LRRKLEELT
DEG_APCC_DBOX_1
0.2778
p.E383K
M14
skin
COSMIC
LRRKLEELT
DEG_APCC_DBOX_1
0.2778
p.N395S
SIDM00878
Breast Carcinoma
GDSC
LRRKLEELT
DEG_APCC_DBOX_1
0.2778
p.N395S
HCC1569
breast
COSMIC
LRRKLEELT
DEG_APCC_DBOX_1
0.2778
p.D379N
DO229224
THCA
ICGC
LRRKLEELT
DEG_APCC_DBOX_1
0.1667
p.T379M
DO41289
UCEC
ICGC
LRRKLEELT
DEG_APCC_DBOX_1
0.1667
p.A378V
DO229232
THCA
ICGC
LRRKLEELT
DEG_APCC_DBOX_1
0.1389
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Drug responses associated with MLPH mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of LRRKLEELT
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
Q9BV36
Melanophilin
DEG_APCC_DBOX_1
385:393
LRRKLEELT
APC,CDC20,FZR1
0.9665
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