DegronMD: protein-targeted degradation, mutation and drug response to degrons
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BSML
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CGC
Degron:
LWLFRD
Uniprot ID:
P40337
Source protein:
von Hippel-Lindau disease tumor suppressor
Source gene:
VHL
Class:
LIG_APCC_ABBA_1
Location:
116:121
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.7835
ASA_SCORE:
22.7833
COIL:
0.1155
CONS_SCORE:
0.7701
DSS_SCORE:
0.145
HELIX:
0.0052
FCONS_SCORE:
1.311
RIG_SCORE:
0.8385
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.C121R
DO20446
KIRC
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.8301
p.L117Q
DO18711
KIRC
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.7765
p.L117Q
DO233339
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.7765
p.L117P
DO19613
KIRC
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.7582
p.L117P
DO17542
KIRC
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.7582
p.D121Y
TCGA-B8-5163
KIRC
TCGA
LWLFRD
LIG_APCC_ABBA_1
0.7325
p.D121Y
TCGA-CJ-4638
KIRC
TCGA
LWLFRD
LIG_APCC_ABBA_1
0.7325
p.D121Y
DO20022
KIRC
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.7325
p.D121Y
DO18978
KIRC
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.7325
p.D121Y
DO46824
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.7325
p.C121Y
DO47060
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.7087
p.L118F
TCGA-D1-A2G5
UCEC
TCGA
LWLFRD
LIG_APCC_ABBA_1
0.6981
p.L118F
DO40918
UCEC
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6981
p.K118N
DO233320
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6918
p.L117V
DO19278
KIRC
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6765
p.L117V
DO16158
KIRC
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6765
p.L117V
DO47246
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6765
p.L117V
DO232086
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6765
p.L117V
DO233508
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6765
p.E119D
DO233563
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6758
p.W117G
DO232120
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6714
p.Y112C
DO233359
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6667
p.L118P
TCGA-B0-5094
KIRC
TCGA
LWLFRD
LIG_APCC_ABBA_1
0.6471
p.L118P
DO16769
KIRC
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6471
p.L118P
DO232150
RECA
ICGC
LWLFRD
LIG_APCC_ABBA_1
0.6471
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Drug responses associated with VHL mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of LWLFRD
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
P40337
von Hippel-Lindau disease tumor suppressor
LIG_APCC_ABBA_1
116:121
LWLFRD
APC,CDC20,FZR1
0.7835
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