DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
NRNALTSIT
Uniprot ID:
Q6ZN30
Source protein:
Zinc finger protein basonuclin-2
Source gene:
BNC2
Class:
DEG_APCC_DBOX_1
Location:
383:391
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.7927
ASA_SCORE:
95.6556
COIL:
0.8524
CONS_SCORE:
0.314
DSS_SCORE:
0.6515
HELIX:
0.1236
FCONS_SCORE:
0.7416
RIG_SCORE:
0.7013
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.R391H
DO222762
COCA
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.8244
p.R391H
DO233748
GACA
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.8244
p.R391H
DO11842
GBM
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.8244
p.S386C
DO219008
BLCA
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.7541
p.S387C
SK-LU-1
lung
COSMIC
NRNALTSIT
DEG_APCC_DBOX_1
0.7541
p.R389Q
DO49828
PRAD
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.7329
p.R389Q
DO50076
UCEC
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.7329
p.S387Y
DO222875
MELA
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.712
p.V385L
AU565
breast
COSMIC
NRNALTSIT
DEG_APCC_DBOX_1
0.6765
p.T391A
TCGA-AX-A0J1
UCEC
TCGA
NRNALTSIT
DEG_APCC_DBOX_1
0.6028
p.T388A
HCC2998
large_intestine
COSMIC
NRNALTSIT
DEG_APCC_DBOX_1
0.6028
p.T391N
TCGA-60-2714
LUSC
TCGA
NRNALTSIT
DEG_APCC_DBOX_1
0.5944
p.P382R
TCGA-13-0920
OV
TCGA
NRNALTSIT
DEG_APCC_DBOX_1
0.3056
p.N392K
TCGA-AJ-A3EK
UCEC
TCGA
NRNALTSIT
DEG_APCC_DBOX_1
0.3056
p.A396G
DO26015
LUAD
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.3056
p.T382A
NCI-H2110
lung
COSMIC
NRNALTSIT
DEG_APCC_DBOX_1
0.3056
p.R393C
DO228927
COCA
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.2778
p.R393C
DO50076
UCEC
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.2778
p.R393C
DO41903
UCEC
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.2778
p.R393C
DO41331
UCEC
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.2778
p.S395I
DO218923
LUAD
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.2222
p.A395V
NCI-H630
large_intestine
COSMIC
NRNALTSIT
DEG_APCC_DBOX_1
0.2222
p.N397H
DO231043
LUSC
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.1667
p.E398K
TCGA-TQ-A7RW
LGG
TCGA
NRNALTSIT
DEG_APCC_DBOX_1
0.1389
p.R375P
DO44299
CESC
ICGC
NRNALTSIT
DEG_APCC_DBOX_1
0.1111
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Drug responses associated with BNC2 mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of NRNALTSIT
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
Q6ZN30
Zinc finger protein basonuclin-2
DEG_APCC_DBOX_1
383:391
NRNALTSIT
APC,CDC20,FZR1
0.7927
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