DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
RRKRLQELE
Uniprot ID:
O95239
Source protein:
Chromosome-associated kinesin KIF4A
Source gene:
KIF4A
Class:
DEG_APCC_DBOX_1
Location:
598:606
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.7386
ASA_SCORE:
117.4333
COIL:
0.0457
CONS_SCORE:
0.4496
DSS_SCORE:
0.3969
HELIX:
0.9577
FCONS_SCORE:
1.2152
RIG_SCORE:
0.7471
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.R599H
TCGA-DW-7838
KIRP
TCGA
RRKRLQELE
DEG_APCC_DBOX_1
0.8244
p.R599H
DO20815
KIRP
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.8244
p.R598L
DO23428
LINC
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.7316
p.R601C
TCGA-KN-8428
KICH
TCGA
RRKRLQELE
DEG_APCC_DBOX_1
0.719
p.R601C
DO220484
KICH
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.719
p.L602I
TCGA-FU-A3HZ
CESC
TCGA
RRKRLQELE
DEG_APCC_DBOX_1
0.7174
p.L602I
DO6308
CESC
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.7174
p.K600R
TCGA-MI-A75I
LIHC
TCGA
RRKRLQELE
DEG_APCC_DBOX_1
0.6126
p.K600R
DO49712
LIHC
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.6126
p.E606D
DO228952
LICA
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.5647
p.E606Q
TCGA-AJ-A3EL
UCEC
TCGA
RRKRLQELE
DEG_APCC_DBOX_1
0.5633
p.E606Q
DO41542
UCEC
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.5633
p.R597C
TCGA-AX-A0J0
UCEC
TCGA
RRKRLQELE
DEG_APCC_DBOX_1
0.3056
p.R597C
TCGA-BS-A0UF
UCEC
TCGA
RRKRLQELE
DEG_APCC_DBOX_1
0.3056
p.R597C
TCGA-D1-A2G0
UCEC
TCGA
RRKRLQELE
DEG_APCC_DBOX_1
0.3056
p.R597C
DO43049
UCEC
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.3056
p.R597C
DO41133
UCEC
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.3056
p.R597C
DO41488
UCEC
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.3056
p.R597H
SIDM01728
Endometrial Carcinoma
GDSC
RRKRLQELE
DEG_APCC_DBOX_1
0.3056
p.R597H
ACH-000173
Endometrial/Uterine Cancer
CCLE
RRKRLQELE
DEG_APCC_DBOX_1
0.3056
p.S595I
DO229216
THCA
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.25
p.K614N
TCGA-AX-A05Z
UCEC
TCGA
RRKRLQELE
DEG_APCC_DBOX_1
0.2222
p.K614N
DO40884
UCEC
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.2222
p.L594F
DO52492
COCA
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.2222
p.L594F
DO228986
LICA
ICGC
RRKRLQELE
DEG_APCC_DBOX_1
0.2222
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Drug responses associated with KIF4A mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of RRKRLQELE
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
O95239
Chromosome-associated kinesin KIF4A
DEG_APCC_DBOX_1
598:606
RRKRLQELE
APC,CDC20,FZR1
0.7386
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