DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
VKENL
Uniprot ID:
Q7Z417
Source protein:
Nuclear fragile X mental retardation-interacting protein 2
Source gene:
NUFIP2
Class:
DEG_APCC_KENBOX_2
Location:
362:366
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.9985
ASA_SCORE:
97.22
COIL:
0.7614
CONS_SCORE:
0.9502
DSS_SCORE:
0.392
HELIX:
0.2022
FCONS_SCORE:
1.422
RIG_SCORE:
0.7624
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.S374Y
TCGA-EO-A3B0
UCEC
TCGA
VKENL
DEG_APCC_KENBOX_2
0.5556
p.S374Y
DO219773
UCEC
ICGC
VKENL
DEG_APCC_KENBOX_2
0.5556
p.S360N
TCGA-EB-A3Y6
SKCM
TCGA
VKENL
DEG_APCC_KENBOX_2
0.2778
p.S360N
DO38081
SKCM
ICGC
VKENL
DEG_APCC_KENBOX_2
0.2778
p.S360R
DO229026
LICA
ICGC
VKENL
DEG_APCC_KENBOX_2
0.2778
p.Y358D
DO222875
MELA
ICGC
VKENL
DEG_APCC_KENBOX_2
0.2222
p.I370V
SIDM00845
Burkitt's Lymphoma
GDSC
VKENL
DEG_APCC_KENBOX_2
0.2222
p.I370V
SIDM00461
Acute Myeloid Leukemia
GDSC
VKENL
DEG_APCC_KENBOX_2
0.2222
p.I370V
SIDM01519
Head and Neck Carcinoma
GDSC
VKENL
DEG_APCC_KENBOX_2
0.2222
p.I370V
ACH-000786
Lymphoma
CCLE
VKENL
DEG_APCC_KENBOX_2
0.2222
p.N372T
TCGA-EY-A1GD
UCEC
TCGA
VKENL
DEG_APCC_KENBOX_2
0.1667
p.N372T
DO42129
UCEC
ICGC
VKENL
DEG_APCC_KENBOX_2
0.1667
p.N372S
SIDM01397
Melanoma
GDSC
VKENL
DEG_APCC_KENBOX_2
0.1667
p.S373F
TCGA-CV-A45U
HNSC
TCGA
VKENL
DEG_APCC_KENBOX_2
0.1389
p.S373F
DO52057
HNSC
ICGC
VKENL
DEG_APCC_KENBOX_2
0.1389
p.P354L
TCGA-EE-A3AA
SKCM
TCGA
VKENL
DEG_APCC_KENBOX_2
0.1111
p.P354L
DO222632
MELA
ICGC
VKENL
DEG_APCC_KENBOX_2
0.1111
p.P354L
DO37571
SKCM
ICGC
VKENL
DEG_APCC_KENBOX_2
0.1111
p.V353L
TCGA-50-5049
LUAD
TCGA
VKENL
DEG_APCC_KENBOX_2
0.0833
p.V353L
DO23705
LUAD
ICGC
VKENL
DEG_APCC_KENBOX_2
0.0833
p.V353A
SIDM00480
Ovarian Carcinoma
GDSC
VKENL
DEG_APCC_KENBOX_2
0.0833
p.V353A
ACH-000704
Ovarian Cancer
CCLE
VKENL
DEG_APCC_KENBOX_2
0.0833
p.V353A
OAW-42
ovary
COSMIC
VKENL
DEG_APCC_KENBOX_2
0.0833
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Drug responses associated with NUFIP2 mutations
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Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of VKENL
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
Q7Z417
Nuclear fragile X mental retardation-interacting protein 2
DEG_APCC_KENBOX_2
362:366
VKENL
APC,CDC20,FZR1
0.9985
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