DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
DASTGE
Uniprot ID:
A2CJ06
Source protein:
Dystrotelin
Source gene:
DYTN
Class:
DEG_Kelch_Keap1_1
Location:
423:428
E3 ligase:
KEAP1
DEGRON score:
0.9713
ASA_SCORE:
91.5167
COIL:
0.8468
CONS_SCORE:
0.1988
DSS_SCORE:
0.6275
HELIX:
0.1428
FCONS_SCORE:
0.7401
RIG_SCORE:
0.6431
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.A424V
TCGA-AA-A00N
COAD
TCGA
DASTGE
DEG_Kelch_Keap1_1
0.5825
p.A424V
DO9876
COAD
ICGC
DASTGE
DEG_Kelch_Keap1_1
0.5825
p.K432T
TCGA-RD-A7BT
STAD
TCGA
DASTGE
DEG_Kelch_Keap1_1
0.3333
p.K432T
DO50131
STAD
ICGC
DASTGE
DEG_Kelch_Keap1_1
0.3333
p.K418N
TCGA-A5-A0G2
UCEC
TCGA
DASTGE
DEG_Kelch_Keap1_1
0.3056
p.K418N
DO41235
UCEC
ICGC
DASTGE
DEG_Kelch_Keap1_1
0.3056
p.K418N
SIDM01124
Non-Small Cell Lung Carcinoma
GDSC
DASTGE
DEG_Kelch_Keap1_1
0.3056
p.K418N
ACH-000945
Lung Cancer
CCLE
DASTGE
DEG_Kelch_Keap1_1
0.3056
p.K418N
NCI-H650
lung
COSMIC
DASTGE
DEG_Kelch_Keap1_1
0.3056
p.E422G
DO228944
LICA
ICGC
DASTGE
DEG_Kelch_Keap1_1
0.3056
p.P429H
SIDM00047
Non-Small Cell Lung Carcinoma
GDSC
DASTGE
DEG_Kelch_Keap1_1
0.3056
p.P429H
ACH-002102
Lung Cancer
CCLE
DASTGE
DEG_Kelch_Keap1_1
0.3056
p.P429H
EMC-BAC-2
lung
COSMIC
DASTGE
DEG_Kelch_Keap1_1
0.3056
p.T421A
SIDM00114
Non-Small Cell Lung Carcinoma
GDSC
DASTGE
DEG_Kelch_Keap1_1
0.2778
p.T421A
H513
pleura
COSMIC
DASTGE
DEG_Kelch_Keap1_1
0.2778
p.P431S
DO222749
MELA
ICGC
DASTGE
DEG_Kelch_Keap1_1
0.25
p.E435V
DO232761
PBCA
ICGC
DASTGE
DEG_Kelch_Keap1_1
0.1389
p.L415S
TCGA-63-A5M9
LUSC
TCGA
DASTGE
DEG_Kelch_Keap1_1
0.1111
p.L415S
DO223726
LUSC
ICGC
DASTGE
DEG_Kelch_Keap1_1
0.1111
p.R438I
TCGA-EO-A22U
UCEC
TCGA
DASTGE
DEG_Kelch_Keap1_1
0.0556
p.R438I
DO43755
UCEC
ICGC
DASTGE
DEG_Kelch_Keap1_1
0.0556
p.D413N
TCGA-Z2-A8RT
SKCM
TCGA
DASTGE
DEG_Kelch_Keap1_1
0.0556
p.D413N
DO51301
SKCM
ICGC
DASTGE
DEG_Kelch_Keap1_1
0.0556
Showing 1 to 23 of 23 entries
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Drug responses associated with DYTN mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of DASTGE
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
A2CJ06
Dystrotelin
DEG_Kelch_Keap1_1
423:428
DASTGE
KEAP1
0.9713
More...
Q9Y5I4
Protocadherin alpha-C2
DEG_Kelch_Keap1_1
311:316
DASTGE
KEAP1
0.9597
More...
Showing 1 to 2 of 2 entries
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