DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
HKENT
Uniprot ID:
P05546
Source protein:
Heparin cofactor 2
Source gene:
SERPIND1
Class:
DEG_APCC_KENBOX_2
Location:
60:64
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.6429
ASA_SCORE:
95.44
COIL:
0.7808
CONS_SCORE:
0.2899
DSS_SCORE:
0.4538
HELIX:
0.1354
FCONS_SCORE:
0.9682
RIG_SCORE:
0.7206
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.E62K
TCGA-D3-A8GM
SKCM
TCGA
HKENT
DEG_APCC_KENBOX_2
0.7022
p.E62K
TCGA-Z2-AA3V
SKCM
TCGA
HKENT
DEG_APCC_KENBOX_2
0.7022
p.E62K
DO50288
SKCM
ICGC
HKENT
DEG_APCC_KENBOX_2
0.7022
p.E62K
DO51303
SKCM
ICGC
HKENT
DEG_APCC_KENBOX_2
0.7022
p.V65I
ACH-002647
Gastric Cancer
CCLE
HKENT
DEG_APCC_KENBOX_2
0.3056
p.N67D
TCGA-EY-A1G8
UCEC
TCGA
HKENT
DEG_APCC_KENBOX_2
0.25
p.N67D
DO43578
UCEC
ICGC
HKENT
DEG_APCC_KENBOX_2
0.25
p.D68E
TCGA-18-3409
LUSC
TCGA
HKENT
DEG_APCC_KENBOX_2
0.2222
p.D68E
DO26444
LUSC
ICGC
HKENT
DEG_APCC_KENBOX_2
0.2222
p.D68N
DO229459
SKCA
ICGC
HKENT
DEG_APCC_KENBOX_2
0.2222
p.L55R
ACH-001991
Primary
CCLE
HKENT
DEG_APCC_KENBOX_2
0.1944
p.P53A
ACH-001057
Lymphoma
CCLE
HKENT
DEG_APCC_KENBOX_2
0.1389
p.E72Q
TCGA-DK-A3IS
BLCA
TCGA
HKENT
DEG_APCC_KENBOX_2
0.1111
p.E72Q
DO566
BLCA
ICGC
HKENT
DEG_APCC_KENBOX_2
0.1111
p.G73E
DO220857
MELA
ICGC
HKENT
DEG_APCC_KENBOX_2
0.0833
p.E74K
TCGA-YG-AA3N
SKCM
TCGA
HKENT
DEG_APCC_KENBOX_2
0.0556
p.E74K
DO51298
SKCM
ICGC
HKENT
DEG_APCC_KENBOX_2
0.0556
Showing 1 to 17 of 17 entries
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Drug responses associated with SERPIND1 mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
No data available in table
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All proteins holding degron of HKENT
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
P05546
Heparin cofactor 2
DEG_APCC_KENBOX_2
60:64
HKENT
APC,CDC20,FZR1
0.6429
More...
Q86VD1
MORC family CW-type zinc finger protein 1
DEG_APCC_KENBOX_2
588:592
HKENT
APC,CDC20,FZR1
0.7009
More...
Showing 1 to 2 of 2 entries
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