DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
HKENT
Uniprot ID:
Q86VD1
Source protein:
MORC family CW-type zinc finger protein 1
Source gene:
MORC1
Class:
DEG_APCC_KENBOX_2
Location:
588:592
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.7009
ASA_SCORE:
111.92
COIL:
0.6582
CONS_SCORE:
0.374
DSS_SCORE:
0.3911
HELIX:
0.3286
FCONS_SCORE:
1.008
RIG_SCORE:
0.7492
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.H588N
TCGA-51-4079
LUSC
TCGA
HKENT
DEG_APCC_KENBOX_2
0.6312
p.H588N
DO26437
LUSC
ICGC
HKENT
DEG_APCC_KENBOX_2
0.6312
p.K596I
TCGA-FD-A5C0
BLCA
TCGA
HKENT
DEG_APCC_KENBOX_2
0.3333
p.K596I
DO44046
BLCA
ICGC
HKENT
DEG_APCC_KENBOX_2
0.3333
p.S596G
ACH-000943
Colon/Colorectal Cancer
CCLE
HKENT
DEG_APCC_KENBOX_2
0.3333
p.S596G
RKO
large_intestine
COSMIC
HKENT
DEG_APCC_KENBOX_2
0.3333
p.A595V
M059J
central_nervous_system
COSMIC
HKENT
DEG_APCC_KENBOX_2
0.25
p.L584I
SIDM00598
Squamous Cell Lung Carcinoma
GDSC
HKENT
DEG_APCC_KENBOX_2
0.2222
p.L584I
ACH-000843
Lung Cancer
CCLE
HKENT
DEG_APCC_KENBOX_2
0.2222
p.L584I
HARA
lung
COSMIC
HKENT
DEG_APCC_KENBOX_2
0.2222
p.D582E
ACH-001618
Leukemia
CCLE
HKENT
DEG_APCC_KENBOX_2
0.1667
p.S581F
TCGA-FS-A1ZK
SKCM
TCGA
HKENT
DEG_APCC_KENBOX_2
0.1389
p.S581F
DO220852
MELA
ICGC
HKENT
DEG_APCC_KENBOX_2
0.1389
p.S581F
DO37474
SKCM
ICGC
HKENT
DEG_APCC_KENBOX_2
0.1389
p.G601V
DO231124
LUSC
ICGC
HKENT
DEG_APCC_KENBOX_2
0.0833
Showing 1 to 15 of 15 entries
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Drug responses associated with MORC1 mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
No data available in table
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All proteins holding degron of HKENT
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
P05546
Heparin cofactor 2
DEG_APCC_KENBOX_2
60:64
HKENT
APC,CDC20,FZR1
0.6429
More...
Q86VD1
MORC family CW-type zinc finger protein 1
DEG_APCC_KENBOX_2
588:592
HKENT
APC,CDC20,FZR1
0.7009
More...
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