DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
DKEND
Uniprot ID:
P49321
Source protein:
Nuclear autoantigenic sperm protein
Source gene:
NASP
Class:
DEG_APCC_KENBOX_2
Location:
484:488
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.9718
ASA_SCORE:
113.6
COIL:
0.6928
CONS_SCORE:
0.4029
DSS_SCORE:
0.8919
HELIX:
0.296
FCONS_SCORE:
1.1615
RIG_SCORE:
0.5919
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.E486D
SIDM00118
Colorectal Carcinoma
GDSC
DKEND
DEG_APCC_KENBOX_2
0.6758
p.E486D
ACH-001081
Colon/Colorectal Cancer
CCLE
DKEND
DEG_APCC_KENBOX_2
0.6758
p.E486D
HCC2998
large_intestine
COSMIC
DKEND
DEG_APCC_KENBOX_2
0.6758
p.S480L
TCGA-E2-A15S
BRCA
TCGA
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
DO5597
BRCA
ICGC
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
SIDM00551
Esophageal Squamous Cell Carcinoma
GDSC
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
SIDM00486
Squamous Cell Lung Carcinoma
GDSC
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
SIDM00580
Acute Myeloid Leukemia
GDSC
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
ACH-000168
Leukemia
CCLE
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
ACH-000563
Lung Cancer
CCLE
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
ACH-002263
Esophageal Cancer
CCLE
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
ACH-002785
Unknown
CCLE
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
EBC-1
lung
COSMIC
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
KYSE-220
oesophagus
COSMIC
DKEND
DEG_APCC_KENBOX_2
0.6667
p.S480L
NOMO-1
haematopoietic_and_lymphoid_tissue
COSMIC
DKEND
DEG_APCC_KENBOX_2
0.6667
p.A480T
MOLT-4
haematopoietic_and_lymphoid_tissue
COSMIC
DKEND
DEG_APCC_KENBOX_2
0.6667
p.D483H
TCGA-DD-AAC8
LIHC
TCGA
DKEND
DEG_APCC_KENBOX_2
0.3056
p.D483H
DO52193
LIHC
ICGC
DKEND
DEG_APCC_KENBOX_2
0.3056
p.E478D
DO233293
NACA
ICGC
DKEND
DEG_APCC_KENBOX_2
0.1667
Showing 1 to 19 of 19 entries
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Drug responses associated with NASP mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of DKEND
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
P30305
M-phase inducer phosphatase 2
DEG_APCC_KENBOX_2
191:195
DKEND
APC,CDC20,FZR1
0.9928
More...
P49321
Nuclear autoantigenic sperm protein
DEG_APCC_KENBOX_2
484:488
DKEND
APC,CDC20,FZR1
0.9718
More...
Q9BZF1
Oxysterol-binding protein-related protein 8
DEG_APCC_KENBOX_2
332:336
DKEND
APC,CDC20,FZR1
0.9813
More...
Showing 1 to 3 of 3 entries
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