DegronMD: protein-targeted degradation, mutation and drug response to degrons
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BSML
CPH
CGC
Degron:
NKENT
Uniprot ID:
Q9NQ76
Source protein:
Matrix extracellular phosphoglycoprotein
Source gene:
MEPE
Class:
DEG_APCC_KENBOX_2
Location:
104:108
E3 ligase:
APC,CDC20,FZR1
DEGRON score:
0.9952
ASA_SCORE:
91.8
COIL:
0.6648
CONS_SCORE:
0.5976
DSS_SCORE:
0.498
HELIX:
0.2798
FCONS_SCORE:
1.3092
RIG_SCORE:
0.6739
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.N107I
DO222843
MELA
ICGC
NKENT
DEG_APCC_KENBOX_2
0.728
p.D107N
DO51298
SKCM
ICGC
NKENT
DEG_APCC_KENBOX_2
0.6932
p.E106D
TCGA-A5-A2K5
UCEC
TCGA
NKENT
DEG_APCC_KENBOX_2
0.6758
p.E106D
TCGA-BS-A0UV
UCEC
TCGA
NKENT
DEG_APCC_KENBOX_2
0.6758
p.T108S
TCGA-50-6593
LUAD
TCGA
NKENT
DEG_APCC_KENBOX_2
0.6005
p.T108S
DO24100
LUAD
ICGC
NKENT
DEG_APCC_KENBOX_2
0.6005
p.N104D
ACH-002317
Leukemia
CCLE
NKENT
DEG_APCC_KENBOX_2
0.5821
p.N104D
YT
haematopoietic_and_lymphoid_tissue
COSMIC
NKENT
DEG_APCC_KENBOX_2
0.5821
p.F102V
DO42280
UCEC
ICGC
NKENT
DEG_APCC_KENBOX_2
0.2778
p.G111C
TCGA-50-5049
LUAD
TCGA
NKENT
DEG_APCC_KENBOX_2
0.25
p.G111C
DO229022
LICA
ICGC
NKENT
DEG_APCC_KENBOX_2
0.25
p.G111C
DO23705
LUAD
ICGC
NKENT
DEG_APCC_KENBOX_2
0.25
p.S101I
TCGA-NC-A5HD
LUSC
TCGA
NKENT
DEG_APCC_KENBOX_2
0.25
p.S101I
DO219184
LUSC
ICGC
NKENT
DEG_APCC_KENBOX_2
0.25
p.K100R
DO36619
READ
ICGC
NKENT
DEG_APCC_KENBOX_2
0.2222
p.E99K
DO10172
COAD
ICGC
NKENT
DEG_APCC_KENBOX_2
0.1944
p.R99S
SIDM00401
Melanoma
GDSC
NKENT
DEG_APCC_KENBOX_2
0.1944
p.R99S
RVH-421
skin
COSMIC
NKENT
DEG_APCC_KENBOX_2
0.1944
p.G113R
SIDM01175
Other Sarcomas
GDSC
NKENT
DEG_APCC_KENBOX_2
0.1944
p.G113R
SW684
soft_tissue
COSMIC
NKENT
DEG_APCC_KENBOX_2
0.1944
p.T97I
DO38111
SKCM
ICGC
NKENT
DEG_APCC_KENBOX_2
0.1389
p.L96M
TCGA-AP-A051
UCEC
TCGA
NKENT
DEG_APCC_KENBOX_2
0.1111
p.L96M
DO42673
UCEC
ICGC
NKENT
DEG_APCC_KENBOX_2
0.1111
p.P118H
TCGA-D3-A2JC
SKCM
TCGA
NKENT
DEG_APCC_KENBOX_2
0.0556
p.P94H
DO47578
SKCM
ICGC
NKENT
DEG_APCC_KENBOX_2
0.0556
Showing 1 to 25 of 27 entries
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Drug responses associated with MEPE mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
No data available in table
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All proteins holding degron of NKENT
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
Q9NQ76
Matrix extracellular phosphoglycoprotein
DEG_APCC_KENBOX_2
104:108
NKENT
APC,CDC20,FZR1
0.9952
More...
Q9NQ76
Matrix extracellular phosphoglycoprotein
DEG_APCC_KENBOX_2
168:172
NKENT
APC,CDC20,FZR1
0.8651
More...
Q8TBY0
Probable RNA-binding protein 46
DEG_APCC_KENBOX_2
310:314
NKENT
APC,CDC20,FZR1
0.8004
More...
O94988
Protein FAM13A
DEG_APCC_KENBOX_2
428:432
NKENT
APC,CDC20,FZR1
0.9473
More...
Showing 1 to 4 of 4 entries
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