VIS ID | Virus | Ensembl ID | Gene Type | Target Gene | Oncogene | Tumor Suppressor Gene | NCBI ID | Uniprot ID |
---|---|---|---|---|---|---|---|---|
TVIS10016573 | HBV | ENSG00000102468.11 | protein_coding | HTR2A | No | No | 3356 | P28223 |
TVIS44041305 | HTLV-1 | ENSG00000102468.11 | protein_coding | HTR2A | No | No | 3356 | P28223 |
Target Gene Table
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TCGA Plot Options
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Drug Information
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Gene | HTR2A |
---|---|
DrugBank ID | DB06016 |
Drug Name | Cariprazine |
Target ID | BE0000451 |
UniProt ID | P28223 |
Regulation Type | antagonist |
PubMed IDs | 26510944; 26956157 |
Citations | McCormack PL: Cariprazine: First Global Approval. Drugs. 2015 Nov;75(17):2035-43. doi: 10.1007/s40265-015-0494-7.@@Stahl SM: Mechanism of action of cariprazine. CNS Spectr. 2016 Apr;21(2):123-7. doi: 10.1017/S1092852916000043. Epub 2016 Mar 9. |
Groups | Approved; Investigational |
Direct Classification | Phenylpiperazines |
SMILES | CN(C)C(=O)N[C@H]1CC[C@H](CCN2CCN(CC2)C2=C(Cl)C(Cl)=CC=C2)CC1 |
Pathways | |
PharmGKB | |
ChEMBL | CHEMBL2028019 |