DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
PITTT
Uniprot ID:
Q9NY46
Source protein:
Sodium channel protein type 3 subunit alpha
Source gene:
SCN3A
Class:
DEG_SPOP_SBC_1
Location:
1890:1894
E3 ligase:
SPOP
DEGRON score:
0.9728
ASA_SCORE:
62.94
COIL:
0.7704
CONS_SCORE:
0.3332
DSS_SCORE:
0.4179
HELIX:
0.116
FCONS_SCORE:
1.0443
RIG_SCORE:
0.7964
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.T1893I
TCGA-W3-A828
SKCM
TCGA
PITTT
DEG_SPOP_SBC_1
0.8189
p.T1893I
DO51273
SKCM
ICGC
PITTT
DEG_SPOP_SBC_1
0.8189
p.T1893I
SIDM00581
Glioblastoma
GDSC
PITTT
DEG_SPOP_SBC_1
0.8189
p.T1893I
ACH-000738
Brain Cancer
CCLE
PITTT
DEG_SPOP_SBC_1
0.8189
p.T1893I
GB-1
central_nervous_system
COSMIC
PITTT
DEG_SPOP_SBC_1
0.8189
p.D1898H
DO51632
CESC
ICGC
PITTT
DEG_SPOP_SBC_1
0.3333
p.G1885R
DO222420
MELA
ICGC
PITTT
DEG_SPOP_SBC_1
0.3056
p.M1895I
DO218847
SKCA
ICGC
PITTT
DEG_SPOP_SBC_1
0.3056
p.K1896M
NCI-H1436
lung
COSMIC
PITTT
DEG_SPOP_SBC_1
0.2778
p.R1897H
TCGA-AA-3977
COAD
TCGA
PITTT
DEG_SPOP_SBC_1
0.25
p.R1897H
TCGA-CG-4460
STAD
TCGA
PITTT
DEG_SPOP_SBC_1
0.25
p.R1897H
SIDM00491
Thyroid Gland Carcinoma
GDSC
PITTT
DEG_SPOP_SBC_1
0.25
p.R1897H
ACH-001443
Thyroid Cancer
CCLE
PITTT
DEG_SPOP_SBC_1
0.25
p.R1897H
ASH-3
thyroid
COSMIC
PITTT
DEG_SPOP_SBC_1
0.25
p.R1897C
SIDM00890
Melanoma
GDSC
PITTT
DEG_SPOP_SBC_1
0.25
p.R1897C
ACH-000580
Skin Cancer
CCLE
PITTT
DEG_SPOP_SBC_1
0.25
p.R1897C
C32
skin
COSMIC
PITTT
DEG_SPOP_SBC_1
0.25
p.K1899T
THP-1
haematopoietic_and_lymphoid_tissue
COSMIC
PITTT
DEG_SPOP_SBC_1
0.1944
p.E1900Q
SIDM00995
Other Solid Cancers
GDSC
PITTT
DEG_SPOP_SBC_1
0.1667
p.E1900Q
ACH-001328
Skin Cancer
CCLE
PITTT
DEG_SPOP_SBC_1
0.1667
p.E1900Q
A431
skin
COSMIC
PITTT
DEG_SPOP_SBC_1
0.1667
p.N1882K
TCGA-17-Z028
LUAD
TCGA
PITTT
DEG_SPOP_SBC_1
0.1111
p.S1881L
TCGA-A5-A0G2
UCEC
TCGA
PITTT
DEG_SPOP_SBC_1
0.0833
p.S1881L
DO41235
UCEC
ICGC
PITTT
DEG_SPOP_SBC_1
0.0833
p.S1881P
TCGA-A5-A1OF
UCEC
TCGA
PITTT
DEG_SPOP_SBC_1
0.0833
Showing 1 to 25 of 34 entries
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Drug responses associated with SCN3A mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of PITTT
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
P27338
Amine oxidase [flavin-containing] B
DEG_SPOP_SBC_1
476:480
PITTT
SPOP
0.8811
More...
A5YKK6
CCR4-NOT transcription complex subunit 1
DEG_SPOP_SBC_1
1331:1335
PITTT
SPOP
0.6964
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
1441:1445
PITTT
SPOP
0.7527
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
1668:1672
PITTT
SPOP
0.5757
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
1684:1688
PITTT
SPOP
0.7501
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
1708:1712
PITTT
SPOP
0.5209
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
1900:1904
PITTT
SPOP
0.9006
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
1923:1927
PITTT
SPOP
0.9531
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
1946:1950
PITTT
SPOP
0.9842
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
1969:1973
PITTT
SPOP
0.9854
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
1992:1996
PITTT
SPOP
0.9953
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2015:2019
PITTT
SPOP
0.9735
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2038:2042
PITTT
SPOP
0.9863
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2061:2065
PITTT
SPOP
0.9919
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2084:2088
PITTT
SPOP
0.9675
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2107:2111
PITTT
SPOP
0.9639
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2130:2134
PITTT
SPOP
0.9712
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2153:2157
PITTT
SPOP
0.9102
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2176:2180
PITTT
SPOP
0.9799
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2199:2203
PITTT
SPOP
0.9635
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2222:2226
PITTT
SPOP
0.9973
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2245:2249
PITTT
SPOP
0.9971
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2268:2272
PITTT
SPOP
0.9967
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2291:2295
PITTT
SPOP
0.9686
More...
Q02817
Mucin-2
DEG_SPOP_SBC_1
2314:2318
PITTT
SPOP
0.9855
More...
Showing 1 to 25 of 119 entries
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