DegronMD: protein-targeted degradation, mutation and drug response to degrons
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BSML
CPH
CGC
Degron:
AKSSS
Uniprot ID:
Q9Y692
Source protein:
Glucocorticoid modulatory element-binding protein 1
Source gene:
GMEB1
Class:
DEG_SPOP_SBC_1
Location:
455:459
E3 ligase:
SPOP
DEGRON score:
0.8751
ASA_SCORE:
81.94
COIL:
0.8584
CONS_SCORE:
0.2295
DSS_SCORE:
0.3577
HELIX:
0.0658
FCONS_SCORE:
0.8363
RIG_SCORE:
0.6205
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.H456Q
DO5493
BRCA
ICGC
AKSSS
DEG_SPOP_SBC_1
0.7582
p.S458N
SIDM00845
Burkitt's Lymphoma
GDSC
AKSSS
DEG_SPOP_SBC_1
0.7069
p.S458N
SIDM00461
Acute Myeloid Leukemia
GDSC
AKSSS
DEG_SPOP_SBC_1
0.7069
p.S458N
SIDM01519
Head and Neck Carcinoma
GDSC
AKSSS
DEG_SPOP_SBC_1
0.7069
p.K456N
SIDM00548
Squamous Cell Lung Carcinoma
GDSC
AKSSS
DEG_SPOP_SBC_1
0.5806
p.K456N
LK-2
lung
COSMIC
AKSSS
DEG_SPOP_SBC_1
0.5806
p.T462P
TCGA-BT-A42C
BLCA
TCGA
AKSSS
DEG_SPOP_SBC_1
0.25
p.T452P
DO49725
BLCA
ICGC
AKSSS
DEG_SPOP_SBC_1
0.25
p.A462V
DO52630
BOCA
ICGC
AKSSS
DEG_SPOP_SBC_1
0.25
p.H466Q
TCGA-E2-A1B6
BRCA
TCGA
AKSSS
DEG_SPOP_SBC_1
0.1389
p.S448I
DO229036
LICA
ICGC
AKSSS
DEG_SPOP_SBC_1
0.1389
p.S448N
ACH-000992
Head and Neck Cancer
CCLE
AKSSS
DEG_SPOP_SBC_1
0.1389
p.R447S
TCGA-AX-A2HC
UCEC
TCGA
AKSSS
DEG_SPOP_SBC_1
0.1111
p.R447H
TCGA-EA-A3HS
CESC
TCGA
AKSSS
DEG_SPOP_SBC_1
0.1111
p.R447H
SIDM00828
Other Sarcomas
GDSC
AKSSS
DEG_SPOP_SBC_1
0.1111
p.R447H
SIDM00500
Colorectal Carcinoma
GDSC
AKSSS
DEG_SPOP_SBC_1
0.1111
p.R447H
HT-1080
soft_tissue
COSMIC
AKSSS
DEG_SPOP_SBC_1
0.1111
p.K446N
DO50917
LICA
ICGC
AKSSS
DEG_SPOP_SBC_1
0.0833
p.K446N
ACH-000769
Lung Cancer
CCLE
AKSSS
DEG_SPOP_SBC_1
0.0833
p.K446N
LK-2
lung
COSMIC
AKSSS
DEG_SPOP_SBC_1
0.0833
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Drug responses associated with GMEB1 mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of AKSSS
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
O94762
ATP-dependent DNA helicase Q5
DEG_SPOP_SBC_1
732:736
AKSSS
SPOP
0.7563
More...
P25440
Bromodomain-containing protein 2
DEG_SPOP_SBC_1
474:478
AKSSS
SPOP
0.6808
More...
O60885
Bromodomain-containing protein 4
DEG_SPOP_SBC_1
1217:1221
AKSSS
SPOP
0.9576
More...
O14647
Chromodomain-helicase-DNA-binding protein 2
DEG_SPOP_SBC_1
1432:1436
AKSSS
SPOP
0.9644
More...
Q9NYV4
Cyclin-dependent kinase 12
DEG_SPOP_SBC_1
167:171
AKSSS
SPOP
0.989
More...
Q9Y692
Glucocorticoid modulatory element-binding protein 1
DEG_SPOP_SBC_1
455:459
AKSSS
SPOP
0.8751
More...
Q9P2N6
KAT8 regulatory NSL complex subunit 3
DEG_SPOP_SBC_1
698:702
AKSSS
SPOP
0.9382
More...
Q2TAC6
Kinesin-like protein KIF19
DEG_SPOP_SBC_1
720:724
AKSSS
SPOP
0.9422
More...
Q96PV6
Leukocyte receptor cluster member 8
DEG_SPOP_SBC_1
59:63
AKSSS
SPOP
0.9898
More...
Q8NEY1
Neuron navigator 1
DEG_SPOP_SBC_1
677:681
AKSSS
SPOP
0.9854
More...
Q5SYE7
NHS-like protein 1
DEG_SPOP_SBC_1
1146:1150
AKSSS
SPOP
0.9831
More...
Q6P4R8
Nuclear factor related to kappa-B-binding protein
DEG_SPOP_SBC_1
755:759
AKSSS
SPOP
0.5292
More...
Q14693
Phosphatidate phosphatase LPIN1
DEG_SPOP_SBC_1
282:286
AKSSS
SPOP
0.9674
More...
Q96BN6
Primary cilium assembly protein FAM149B1
DEG_SPOP_SBC_1
203:207
AKSSS
SPOP
0.9219
More...
Q6PRD1
Probable G-protein coupled receptor 179
DEG_SPOP_SBC_1
906:910
AKSSS
SPOP
0.9545
More...
Q5VWN6
Protein TASOR 2
DEG_SPOP_SBC_1
1165:1169
AKSSS
SPOP
0.9726
More...
A6NCF6
Putative MAGE domain-containing protein MAGEA13P
DEG_SPOP_SBC_1
332:336
AKSSS
SPOP
0.9368
More...
O95294
RasGAP-activating-like protein 1
DEG_SPOP_SBC_1
2:6
AKSSS
SPOP
0.7406
More...
Q9NWH9
SAFB-like transcription modulator
DEG_SPOP_SBC_1
351:355
AKSSS
SPOP
0.9894
More...
Q6ZVL6
UPF0606 protein KIAA1549L
DEG_SPOP_SBC_1
676:680
AKSSS
SPOP
0.9984
More...
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