DegronMD: protein-targeted degradation, mutation and drug response to degrons
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BSML
CPH
CGC
Degron:
AATTT
Uniprot ID:
O60907
Source protein:
F-box-like/WD repeat-containing protein TBL1X
Source gene:
TBL1X
Class:
DEG_SPOP_SBC_1
Location:
174:178
E3 ligase:
SPOP
DEGRON score:
0.6842
ASA_SCORE:
79.2
COIL:
0.652
CONS_SCORE:
0.2565
DSS_SCORE:
0.4859
HELIX:
0.274
FCONS_SCORE:
0.8896
RIG_SCORE:
0.6828
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.R178W
DO35442
PACA
ICGC
AATTT
DEG_SPOP_SBC_1
0.8634
p.R178Q
DO10694
COAD
ICGC
AATTT
DEG_SPOP_SBC_1
0.7329
p.L177I
DO37782
SKCM
ICGC
AATTT
DEG_SPOP_SBC_1
0.7174
p.T175A
DO6466
CLLE
ICGC
AATTT
DEG_SPOP_SBC_1
0.7139
p.G179V
DO229019
LICA
ICGC
AATTT
DEG_SPOP_SBC_1
0.3056
p.G179V
DO229028
LICA
ICGC
AATTT
DEG_SPOP_SBC_1
0.3056
p.H180R
DO42472
UCEC
ICGC
AATTT
DEG_SPOP_SBC_1
0.2778
p.V182I
TCGA-12-0692
GBM
TCGA
AATTT
DEG_SPOP_SBC_1
0.2222
p.A170S
TCGA-55-A492
LUAD
TCGA
AATTT
DEG_SPOP_SBC_1
0.2222
p.S183P
ACH-000993
Endometrial/Uterine Cancer
CCLE
AATTT
DEG_SPOP_SBC_1
0.1944
p.I186M
DO231602
LINC
ICGC
AATTT
DEG_SPOP_SBC_1
0.1111
p.A165V
SIDM00951
T-Lymphoblastic Leukemia
GDSC
AATTT
DEG_SPOP_SBC_1
0.0833
p.A164V
TCGA-5M-AAT6
COAD
TCGA
AATTT
DEG_SPOP_SBC_1
0.0556
p.S188L
TCGA-EO-A22U
UCEC
TCGA
AATTT
DEG_SPOP_SBC_1
0.0556
Showing 1 to 14 of 14 entries
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Drug responses associated with TBL1X mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
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All proteins holding degron of AATTT
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
Q9UKB5
Adherens junction-associated protein 1
DEG_SPOP_SBC_1
217:221
AATTT
SPOP
0.9943
More...
O60641
Clathrin coat assembly protein AP180
DEG_SPOP_SBC_1
542:546
AATTT
SPOP
0.611
More...
O60907
F-box-like/WD repeat-containing protein TBL1X
DEG_SPOP_SBC_1
174:178
AATTT
SPOP
0.6842
More...
Q8N3X1
Formin-binding protein 4
DEG_SPOP_SBC_1
53:57
AATTT
SPOP
0.704
More...
Q6ZRS2
Helicase SRCAP
DEG_SPOP_SBC_1
1143:1147
AATTT
SPOP
0.8846
More...
P55318
Hepatocyte nuclear factor 3-gamma
DEG_SPOP_SBC_1
226:230
AATTT
SPOP
0.9972
More...
Q86Z02
Homeodomain-interacting protein kinase 1
DEG_SPOP_SBC_1
156:160
AATTT
SPOP
0.6639
More...
Q96N19
Integral membrane protein GPR137
DEG_SPOP_SBC_1
349:353
AATTT
SPOP
0.882
More...
Q9HCJ2
Leucine-rich repeat-containing protein 4C
DEG_SPOP_SBC_1
445:449
AATTT
SPOP
0.8689
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Q8IZL2
Mastermind-like protein 2
DEG_SPOP_SBC_1
99:103
AATTT
SPOP
0.8339
More...
Q9HC84
Mucin-5B
DEG_SPOP_SBC_1
2999:3003
AATTT
SPOP
0.9608
More...
Q9HC84
Mucin-5B
DEG_SPOP_SBC_1
3141:3145
AATTT
SPOP
0.995
More...
Q9HC84
Mucin-5B
DEG_SPOP_SBC_1
4398:4402
AATTT
SPOP
0.999
More...
Q8WY41
Nanos homolog 1
DEG_SPOP_SBC_1
172:176
AATTT
SPOP
0.8881
More...
P35658
Nuclear pore complex protein Nup214
DEG_SPOP_SBC_1
1824:1828
AATTT
SPOP
0.6214
More...
Q5PRF9
Protein Smaug homolog 2
DEG_SPOP_SBC_1
403:407
AATTT
SPOP
0.9499
More...
Q8IYB3
Serine/arginine repetitive matrix protein 1
DEG_SPOP_SBC_1
852:856
AATTT
SPOP
0.9784
More...
Q9H4A3
Serine/threonine-protein kinase WNK1
DEG_SPOP_SBC_1
69:73
AATTT
SPOP
0.9948
More...
Showing 1 to 18 of 18 entries
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