DegronMD: protein-targeted degradation, mutation and drug response to degrons
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Degron:
AVSSS
Uniprot ID:
Q15714
Source protein:
TSC22 domain family protein 1
Source gene:
TSC22D1
Class:
DEG_SPOP_SBC_1
Location:
279:283
E3 ligase:
SPOP
DEGRON score:
0.9984
ASA_SCORE:
79
COIL:
0.9406
CONS_SCORE:
0.3555
DSS_SCORE:
0.5226
HELIX:
0.026
FCONS_SCORE:
1.017
RIG_SCORE:
0.6122
Degron related mutations and impact score
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Mutation
Sample
Cancer
Dataset
Degron
Degron class
Impact score
p.S282F
SIDM01156
Small Cell Lung Carcinoma
GDSC
AVSSS
DEG_SPOP_SBC_1
0.7982
p.S282F
ACH-000890
Lung Cancer
CCLE
AVSSS
DEG_SPOP_SBC_1
0.7982
p.S282F
SW1271
lung
COSMIC
AVSSS
DEG_SPOP_SBC_1
0.7982
p.S281L
TCGA-VS-A94X
CESC
TCGA
AVSSS
DEG_SPOP_SBC_1
0.7667
p.S281L
DO51632
CESC
ICGC
AVSSS
DEG_SPOP_SBC_1
0.7667
p.P286L
DO218860
SKCA
ICGC
AVSSS
DEG_SPOP_SBC_1
0.25
p.V289A
TCGA-AG-A002
READ
TCGA
AVSSS
DEG_SPOP_SBC_1
0.1667
p.V289G
SIDM00607
Glioblastoma
GDSC
AVSSS
DEG_SPOP_SBC_1
0.1667
p.V289G
ACH-000622
Brain Cancer
CCLE
AVSSS
DEG_SPOP_SBC_1
0.1667
p.V289G
KNS-42
central_nervous_system
COSMIC
AVSSS
DEG_SPOP_SBC_1
0.1667
p.N292I
DO222884
COCA
ICGC
AVSSS
DEG_SPOP_SBC_1
0.0833
p.D269E
DO228976
LICA
ICGC
AVSSS
DEG_SPOP_SBC_1
0.0556
Showing 1 to 12 of 12 entries
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Drug responses associated with TSC22D1 mutations
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Sample
Cancer
Mutation (In Degron?)
Dataset
Drug
IC50
No data available in table
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All proteins holding degron of AVSSS
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Uniprot ID
Source protein
Degron class
Location
Hit
E3 ligase
Degron score
Detail
Q0VDD7
Break repair meiotic recombinase recruitment factor 1
DEG_SPOP_SBC_1
66:70
AVSSS
SPOP
0.9837
More...
Q9HCK8
Chromodomain-helicase-DNA-binding protein 8
DEG_SPOP_SBC_1
142:146
AVSSS
SPOP
0.9881
More...
Q8IZA0
Dyslexia-associated protein KIAA0319-like protein
DEG_SPOP_SBC_1
173:177
AVSSS
SPOP
0.8972
More...
P17483
Homeobox protein Hox-B4
DEG_SPOP_SBC_1
112:116
AVSSS
SPOP
0.9569
More...
P32242
Homeobox protein OTX1
DEG_SPOP_SBC_1
131:135
AVSSS
SPOP
0.9911
More...
Q9Y4X4
Krueppel-like factor 12
DEG_SPOP_SBC_1
95:99
AVSSS
SPOP
0.9994
More...
P43358
Melanoma-associated antigen 4
DEG_SPOP_SBC_1
39:43
AVSSS
SPOP
0.8472
More...
Q96JE9
Microtubule-associated protein 6
DEG_SPOP_SBC_1
296:300
AVSSS
SPOP
0.8997
More...
P54278
Mismatch repair endonuclease PMS2
DEG_SPOP_SBC_1
474:478
AVSSS
SPOP
0.999
More...
Q685J3
Mucin-17
DEG_SPOP_SBC_1
1491:1495
AVSSS
SPOP
0.9129
More...
Q685J3
Mucin-17
DEG_SPOP_SBC_1
1844:1848
AVSSS
SPOP
0.8391
More...
Q9ULH7
Myocardin-related transcription factor B
DEG_SPOP_SBC_1
437:441
AVSSS
SPOP
0.6865
More...
Q13613
Myotubularin-related protein 1
DEG_SPOP_SBC_1
643:647
AVSSS
SPOP
0.8381
More...
Q8NEY8
Periphilin-1
DEG_SPOP_SBC_1
211:215
AVSSS
SPOP
0.9988
More...
Q96PX9
Pleckstrin homology domain-containing family G member 4B
DEG_SPOP_SBC_1
1174:1178
AVSSS
SPOP
0.7969
More...
Q92562
Polyphosphoinositide phosphatase
DEG_SPOP_SBC_1
753:757
AVSSS
SPOP
0.9974
More...
P84996
Protein ALEX
DEG_SPOP_SBC_1
603:607
AVSSS
SPOP
0.9965
More...
Q9UPA5
Protein bassoon
DEG_SPOP_SBC_1
3392:3396
AVSSS
SPOP
0.8731
More...
Q06455
Protein CBFA2T1
DEG_SPOP_SBC_1
565:569
AVSSS
SPOP
0.9927
More...
P34910
Protein EVI2B
DEG_SPOP_SBC_1
329:333
AVSSS
SPOP
0.9223
More...
Q5U5X8
Protein FAM222A
DEG_SPOP_SBC_1
109:113
AVSSS
SPOP
0.9845
More...
Q68D20
Protein PMS2CL
DEG_SPOP_SBC_1
88:92
AVSSS
SPOP
0.7454
More...
P43359
Putative melanoma-associated antigen 5P
DEG_SPOP_SBC_1
38:42
AVSSS
SPOP
0.8963
More...
Q9NSC2
Sal-like protein 1
DEG_SPOP_SBC_1
369:373
AVSSS
SPOP
0.7672
More...
Q9H2S1
Small conductance calcium-activated potassium channel protein 2
DEG_SPOP_SBC_1
58:62
AVSSS
SPOP
0.5155
More...
Showing 1 to 25 of 35 entries
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