Drug response data for drug treatments from CCLE, GDSC
This table shows the screened drugs for each kinase. A full list of drug response can be accessed here with treated cell lines in CCLE and GDSC.
| Uniprot ID | Gene symbol | Drug | AVG_IC50(uM) | Details |
| P00519 | ABL1 | AZD0530 | 6.5298 | More.. |
| P00519 | ABL1 | Bosutinib | 12.0191 | More.. |
| P00519 | ABL1 | Dasatinib | 16.1154 | More.. |
| P00519 | ABL1 | GNF-2 | 13.9077 | More.. |
| P00519 | ABL1 | HG-5-113-01 | 8.989 | More.. |
| P00519 | ABL1 | Imatinib | 21.287 | More.. |
| P00519 | ABL1 | Nilotinib | 7.0763 | More.. |
| P00519 | ABL1 | Ponatinib | 3.331 | More.. |
| P00519 | ABL1 | Saracatinib | 15.3916 | More.. |
| P36896 | ACVR1B | SB505124 | 87.8055 | More.. |
| Q8NER5 | ACVR1C | SB505124 | 87.8055 | More.. |
| P31749 | AKT1 | A-443654 | 1.6767 | More.. |
| P31749 | AKT1 | Afuresertib | 33.6297 | More.. |
| P31749 | AKT1 | AKT inhibitor VIII | 23.3743 | More.. |
| P31749 | AKT1 | AT13148 | 154.3793 | More.. |
| P31749 | AKT1 | AZD5363 | 49.9909 | More.. |
| P31749 | AKT1 | GSK690693 | 83.2234 | More.. |
| P31749 | AKT1 | Ipatasertib | 76.4042 | More.. |
| P31749 | AKT1 | MK-2206 | 39.732 | More.. |
| P31749 | AKT1 | Uprosertib | 73.4424 | More.. |
| P31751 | AKT2 | A-443654 | 1.6767 | More.. |
| P31751 | AKT2 | Afuresertib | 33.6297 | More.. |
| P31751 | AKT2 | AKT inhibitor VIII | 23.3743 | More.. |
| P31751 | AKT2 | AZD5363 | 49.9909 | More.. |
| P31751 | AKT2 | GSK690693 | 83.2234 | More.. |
| P31751 | AKT2 | MK-2206 | 39.732 | More.. |
| P31751 | AKT2 | Uprosertib | 73.4424 | More.. |
| Q9Y243 | AKT3 | A-443654 | 1.6767 | More.. |
| Q9Y243 | AKT3 | Afuresertib | 33.6297 | More.. |
| Q9Y243 | AKT3 | AKT inhibitor VIII | 23.3743 | More.. |
| Q9Y243 | AKT3 | AZD5363 | 49.9909 | More.. |
| Q9Y243 | AKT3 | GSK690693 | 83.2234 | More.. |
| Q9Y243 | AKT3 | Ipatasertib | 76.4042 | More.. |
| Q9Y243 | AKT3 | Uprosertib | 73.4424 | More.. |
| Q9UM73 | ALK | Alectinib | 54.1968 | More.. |
| Q9UM73 | ALK | Crizotinib | 42.3076 | More.. |
| Q9UM73 | ALK | NVP-TAE684 | 5.7264 | More.. |
| Q9UM73 | ALK | TAE684 | 4.3779 | More.. |
| Q9UM73 | ALK | XMD14-99 | 112.679 | More.. |
| P10398 | ARAF | RAF_9304 | 19.6052 | More.. |
| Q13315 | ATM | CP466722 | 27.5393 | More.. |
| Q13315 | ATM | KU-55933 | 80.0459 | More.. |
| Q13315 | ATM | KU-60019 | 42.0588 | More.. |
| Q13535 | ATR | AZ20 | 5.4367 | More.. |
| Q13535 | ATR | AZD6738 | 20.0217 | More.. |
| Q13535 | ATR | QL-VIII-58 | 1.1799 | More.. |
| Q13535 | ATR | VE-822 | 89.8091 | More.. |
| Q13535 | ATR | VE821 | 178.7814 | More.. |
| O14965 | AURKA | Alisertib | 24.7294 | More.. |
| O14965 | AURKA | CD532 | 2.1329 | More.. |
| O14965 | AURKA | Genentech Cpd 10 | 34.7087 | More.. |
| O14965 | AURKA | GSK1070916 | 17.3597 | More.. |
| O14965 | AURKA | Tozasertib | 23.3222 | More.. |
| O14965 | AURKA | ZM447439 | 20.5756 | More.. |
| Q96GD4 | AURKB | BX795 | 15.6412 | More.. |
| Q96GD4 | AURKB | Genentech Cpd 10 | 34.7087 | More.. |
| Q96GD4 | AURKB | SL0101 | 101.4104 | More.. |
| Q96GD4 | AURKB | Tozasertib | 23.3222 | More.. |
| Q96GD4 | AURKB | ZM447439 | 20.5756 | More.. |
| Q9UQB9 | AURKC | BX795 | 15.6412 | More.. |
| Q9UQB9 | AURKC | GSK1070916 | 17.3597 | More.. |
| Q9UQB9 | AURKC | Tozasertib | 23.3222 | More.. |
| P30530 | AXL | Cabozantinib | 29.0162 | More.. |
| P51813 | BMX | QL-XII-47 | 17.6755 | More.. |
| P51813 | BMX | QL-XII-61 | 77.5985 | More.. |
| P51813 | BMX | WZ-1-84 | 69.5468 | More.. |
| P15056 | BRAF | AZ628 | 14.2459 | More.. |
| P15056 | BRAF | Dabrafenib | 137.306 | More.. |
| P15056 | BRAF | HG6-64-1 | 10.1773 | More.. |
| P15056 | BRAF | PLX-4720 | 121.6819 | More.. |
| P15056 | BRAF | PLX4720 | 7.3756 | More.. |
| P15056 | BRAF | RAF265 | 3.9296 | More.. |
| P15056 | BRAF | RAF_9304 | 19.6052 | More.. |
| P15056 | BRAF | SB590885 | 54.4715 | More.. |
| P25440 | BRD2 | I-BET-762 | 96.7542 | More.. |
| P25440 | BRD2 | JQ1 | 8.7326 | More.. |
| P25440 | BRD2 | OTX015 | 52.6751 | More.. |
| Q15059 | BRD3 | I-BET-762 | 96.7542 | More.. |
| Q15059 | BRD3 | JQ1 | 8.7326 | More.. |
| Q15059 | BRD3 | OTX015 | 52.6751 | More.. |
| O60885 | BRD4 | AZD5153 | 21.9062 | More.. |
| O60885 | BRD4 | I-BET-762 | 96.7542 | More.. |
| O60885 | BRD4 | JQ1 | 8.7326 | More.. |
| O60885 | BRD4 | OTX015 | 52.6751 | More.. |
| O60885 | BRD4 | PFI-1 | 26.0563 | More.. |
| O60885 | BRD4 | RVX-208 | 206.5075 | More.. |
| Q58F21 | BRDT | JQ1 | 8.7326 | More.. |
| Q8IWQ3 | BRSK2 | XMD11-85h | 69.693 | More.. |
| Q06187 | BTK | Ibrutinib | 217.3064 | More.. |
| Q06187 | BTK | LFM-A13 | 129.4564 | More.. |
| Q06187 | BTK | QL-X-138 | 19.5856 | More.. |
| Q06187 | BTK | QL-XII-47 | 17.6755 | More.. |
| Q06187 | BTK | QL-XII-61 | 77.5985 | More.. |
| Q13554 | CAMK2B | XMD15-27 | 130.6499 | More.. |
| P06493 | CDK1 | AT-7519 | 14.5075 | More.. |
| P06493 | CDK1 | CGP-60474 | 0.35 | More.. |
| P06493 | CDK1 | Dinaciclib | 0.4746 | More.. |
| P06493 | CDK1 | RO-3306 | 41.7289 | More.. |
| P24941 | CDK2 | AT-7519 | 14.5075 | More.. |
| P24941 | CDK2 | AZD5438 | 25.9704 | More.. |
| P24941 | CDK2 | CGP-60474 | 0.35 | More.. |
| P24941 | CDK2 | Dinaciclib | 0.4746 | More.. |
| P24941 | CDK2 | MK-8776 | 68.1764 | More.. |
| P24941 | CDK2 | PHA-793887 | 47.3909 | More.. |
| P24941 | CDK2 | Seliciclib | 82.4724 | More.. |
| P24941 | CDK2 | Staurosporine | 0.2727 | More.. |
| P11802 | CDK4 | AT-7519 | 14.5075 | More.. |
| P11802 | CDK4 | CGP-082996 | 28.1048 | More.. |
| P11802 | CDK4 | Palbociclib | 58.5017 | More.. |
| P11802 | CDK4 | PD-0332991 | 7.1325 | More.. |
| P11802 | CDK4 | Ribociclib | 114.6315 | More.. |
| Q00535 | CDK5 | CGP-60474 | 0.35 | More.. |
| Q00535 | CDK5 | Dinaciclib | 0.4746 | More.. |
| Q00535 | CDK5 | PHA-793887 | 47.3909 | More.. |
| Q00534 | CDK6 | AT-7519 | 14.5075 | More.. |
| Q00534 | CDK6 | Palbociclib | 58.5017 | More.. |
| Q00534 | CDK6 | Ribociclib | 114.6315 | More.. |
| P50613 | CDK7 | CGP-60474 | 0.35 | More.. |
| P50613 | CDK7 | PHA-793887 | 47.3909 | More.. |
| P50613 | CDK7 | Seliciclib | 82.4724 | More.. |
| P50613 | CDK7 | THZ-2-102-1 | 7.1882 | More.. |
| P50613 | CDK7 | XMD14-99 | 112.679 | More.. |
| P50750 | CDK9 | AT-7519 | 14.5075 | More.. |
| P50750 | CDK9 | CDK9_5038 | 1.5719 | More.. |
| P50750 | CDK9 | CDK9_5576 | 4.8221 | More.. |
| P50750 | CDK9 | CGP-60474 | 0.35 | More.. |
| P50750 | CDK9 | Dinaciclib | 0.4746 | More.. |
| P50750 | CDK9 | KIN001-270 | 184.9318 | More.. |
| P50750 | CDK9 | Seliciclib | 82.4724 | More.. |
| P50750 | CDK9 | THZ-2-49 | 92.1592 | More.. |
| P50750 | CDK9 | TL-1-85 | 56.8664 | More.. |
| O14757 | CHEK1 | AZD7762 | 3.0365 | More.. |
| O14757 | CHEK1 | MK-8776 | 68.1764 | More.. |
| O14757 | CHEK1 | Wee1 Inhibitor | 29.3482 | More.. |
| O96017 | CHEK2 | AZD7762 | 3.0365 | More.. |
| O96017 | CHEK2 | MK-8776 | 68.1764 | More.. |
| O15111 | CHUK | BMS-345541 | 35.8809 | More.. |
| Q9HAZ1 | CLK4 | PI-103 | 26.7989 | More.. |
| Q96D53 | COQ8B | HG-5-88-01 | 46.5351 | More.. |
| P07333 | CSF1R | GW-2580 | 240.5333 | More.. |
| P07333 | CSF1R | Linifanib | 12.4093 | More.. |
| P07333 | CSF1R | Pazopanib | 44.186 | More.. |
| P07333 | CSF1R | Sunitinib | 34.8767 | More.. |
| P41240 | CSK | Staurosporine | 0.2727 | More.. |
| O43293 | DAPK3 | PI-103 | 26.7989 | More.. |
| Q08345 | DDR1 | QL-XI-92 | 79.5401 | More.. |
| Q9Y463 | DYRK1B | Dyrk1b_0191 | 23.5127 | More.. |
| O00418 | EEF2K | EEF2K Inhibitor, A-484954 | 308.3359 | More.. |
| P00533 | EGFR | Afatinib | 27.0568 | More.. |
| P00533 | EGFR | AST-1306 | 15.1321 | More.. |
| P00533 | EGFR | AZD3759 | 22.5028 | More.. |
| P00533 | EGFR | AZD8931 | 15.4163 | More.. |
| P00533 | EGFR | Cetuximab | 555.4337 | More.. |
| P00533 | EGFR | CI-1033 | 30.3403 | More.. |
| P00533 | EGFR | CUDC-101 | 4.9464 | More.. |
| P00533 | EGFR | Erlotinib | 17.829 | More.. |
| P00533 | EGFR | Foretinib | 7.1741 | More.. |
| P00533 | EGFR | Gefitinib | 21.3428 | More.. |
| P00533 | EGFR | HG-5-88-01 | 46.5351 | More.. |
| P00533 | EGFR | Lapatinib | 42.8605 | More.. |
| P00533 | EGFR | Osimertinib | 11.2143 | More.. |
| P00533 | EGFR | Pelitinib | 20.3063 | More.. |
| P00533 | EGFR | PF-00299804 | 14.8504 | More.. |
| P00533 | EGFR | Sapitinib | 116.1406 | More.. |
| P00533 | EGFR | ZD-6474 | 6.1987 | More.. |
| P29317 | EPHA2 | Dasatinib | 16.1154 | More.. |
| P54760 | EPHB4 | EphB4_9721 | 24.7725 | More.. |
| P54760 | EPHB4 | NVP-BHG712 | 50.631 | More.. |
| P04626 | ERBB2 | Afatinib | 27.0568 | More.. |
| P04626 | ERBB2 | AZD8931 | 15.4163 | More.. |
| P04626 | ERBB2 | CI-1033 | 30.3403 | More.. |
| P04626 | ERBB2 | CP724714 | 97.1386 | More.. |
| P04626 | ERBB2 | CUDC-101 | 4.9464 | More.. |
| P04626 | ERBB2 | Lapatinib | 58.6235 | More.. |
| P04626 | ERBB2 | PF-00299804 | 14.8504 | More.. |
| P04626 | ERBB2 | Sapitinib | 116.1406 | More.. |
| P21860 | ERBB3 | AZD8931 | 15.4163 | More.. |
| P21860 | ERBB3 | Sapitinib | 116.1406 | More.. |
| Q15303 | ERBB4 | AST-1306 | 15.1321 | More.. |
| Q15303 | ERBB4 | CI-1033 | 30.3403 | More.. |
| Q15303 | ERBB4 | PF-00299804 | 14.8504 | More.. |
| P11362 | FGFR1 | AZD4547 | 27.5072 | More.. |
| P11362 | FGFR1 | BIBF-1120 | 44.8965 | More.. |
| P11362 | FGFR1 | Cediranib | 20.4673 | More.. |
| P11362 | FGFR1 | FGFR_3831 | 37.0744 | More.. |
| P11362 | FGFR1 | Foretinib | 7.1741 | More.. |
| P11362 | FGFR1 | PD173074 | 63.625 | More.. |
| P11362 | FGFR1 | Ponatinib | 3.331 | More.. |
| P11362 | FGFR1 | TKI258 | 5.8784 | More.. |
| P21802 | FGFR2 | AZD4547 | 33.1479 | More.. |
| P21802 | FGFR2 | FGFR_3831 | 37.0744 | More.. |
| P21802 | FGFR2 | PD173074 | 63.625 | More.. |
| P22607 | FGFR3 | AZD4547 | 33.1479 | More.. |
| P22607 | FGFR3 | FGFR_3831 | 37.0744 | More.. |
| P22607 | FGFR3 | PD173074 | 63.625 | More.. |
| P22455 | FGFR4 | FGFR_0939 | 12.3685 | More.. |
| P22455 | FGFR4 | FGFR_3831 | 37.0744 | More.. |
| P09769 | FGR | Midostaurin | 2.0639 | More.. |
| P17948 | FLT1 | Cabozantinib | 29.0162 | More.. |
| P17948 | FLT1 | Cediranib | 20.4673 | More.. |
| P17948 | FLT1 | Linifanib | 12.4093 | More.. |
| P17948 | FLT1 | Midostaurin | 2.0639 | More.. |
| P17948 | FLT1 | Tivozanib | 1.6372 | More.. |
| P36888 | FLT3 | Amuvatinib | 83.9825 | More.. |
| P36888 | FLT3 | Cabozantinib | 29.0162 | More.. |
| P36888 | FLT3 | Cediranib | 20.4673 | More.. |
| P36888 | FLT3 | Lestaurtinib | 2.1852 | More.. |
| P36888 | FLT3 | Linifanib | 12.4093 | More.. |
| P36888 | FLT3 | Ponatinib | 3.331 | More.. |
| P36888 | FLT3 | Quizartinib | 11.5942 | More.. |
| P36888 | FLT3 | Sunitinib | 34.8767 | More.. |
| P36888 | FLT3 | WZ3105 | 6.3868 | More.. |
| P35916 | FLT4 | Cabozantinib | 29.0162 | More.. |
| P35916 | FLT4 | Cediranib | 20.4673 | More.. |
| P35916 | FLT4 | Foretinib | 7.1741 | More.. |
| P35916 | FLT4 | Linifanib | 12.4093 | More.. |
| P35916 | FLT4 | Tivozanib | 1.6372 | More.. |
| P35916 | FLT4 | XMD11-85h | 69.693 | More.. |
| P06241 | FYN | A-770041 | 22.6297 | More.. |
| P49840 | GSK3A | CHIR-99021 | 47.8958 | More.. |
| P49840 | GSK3A | SB216763 | 151.019 | More.. |
| P49841 | GSK3B | AZD7969 | 24.4945 | More.. |
| P49841 | GSK3B | CHIR-99021 | 47.8958 | More.. |
| P49841 | GSK3B | KIN001-042 | 103.8196 | More.. |
| P49841 | GSK3B | SB216763 | 151.019 | More.. |
| P49841 | GSK3B | Staurosporine | 0.2727 | More.. |
| Q9H2X6 | HIPK2 | PI-103 | 26.7989 | More.. |
| P08069 | IGF1R | AEW541 | 5.8337 | More.. |
| P08069 | IGF1R | BMS-536924 | 17.8264 | More.. |
| P08069 | IGF1R | BMS-754807 | 6.0629 | More.. |
| P08069 | IGF1R | GSK1904529A | 81.1251 | More.. |
| P08069 | IGF1R | Linsitinib | 57.4734 | More.. |
| P08069 | IGF1R | NVP-ADW742 | 62.6242 | More.. |
| O14920 | IKBKB | BMS-345541 | 35.8809 | More.. |
| O14920 | IKBKB | IMD-0354 | 6.1016 | More.. |
| O14920 | IKBKB | KIN001-260 | 167.3173 | More.. |
| O14920 | IKBKB | TPCA-1 | 60.8845 | More.. |
| P51617 | IRAK1 | WZ3105 | 6.3868 | More.. |
| Q9NWZ3 | IRAK4 | IRAK4_4710 | 209.0796 | More.. |
| Q08881 | ITK | BMS-509744 | 35.1187 | More.. |
| Q08881 | ITK | Staurosporine | 0.2727 | More.. |
| P23458 | JAK1 | AZD1480 | 8.4029 | More.. |
| P23458 | JAK1 | JAK1_3715 | 97.1079 | More.. |
| P23458 | JAK1 | JAK1_8709 | 126.6849 | More.. |
| P23458 | JAK1 | JAK_8517 | 84.3262 | More.. |
| P23458 | JAK1 | Ruxolitinib | 123.5261 | More.. |
| O60674 | JAK2 | AZ960 | 42.5403 | More.. |
| O60674 | JAK2 | AZD1480 | 8.4029 | More.. |
| O60674 | JAK2 | Fedratinib | 31.0534 | More.. |
| O60674 | JAK2 | JAK_8517 | 84.3262 | More.. |
| O60674 | JAK2 | Lestaurtinib | 2.1852 | More.. |
| O60674 | JAK2 | Ruxolitinib | 123.5261 | More.. |
| P52333 | JAK3 | AZ960 | 42.5403 | More.. |
| P52333 | JAK3 | JAK3_7406 | 53.3468 | More.. |
| P52333 | JAK3 | WHI-P97 | 82.5607 | More.. |
| P35968 | KDR | Axitinib | 16.3642 | More.. |
| P35968 | KDR | BIBF-1120 | 44.8965 | More.. |
| P35968 | KDR | Brivanib, BMS-540215 | 117.5343 | More.. |
| P35968 | KDR | Cabozantinib | 29.0162 | More.. |
| P35968 | KDR | Cediranib | 20.4673 | More.. |
| P35968 | KDR | Foretinib | 7.1741 | More.. |
| P35968 | KDR | Linifanib | 12.4093 | More.. |
| P35968 | KDR | Motesanib | 18.9152 | More.. |
| P35968 | KDR | Ponatinib | 3.331 | More.. |
| P35968 | KDR | Sorafenib | 29.6257 | More.. |
| P35968 | KDR | Sunitinib | 34.8767 | More.. |
| P35968 | KDR | Tivozanib | 1.6372 | More.. |
| P10721 | KIT | Amuvatinib | 83.9825 | More.. |
| P10721 | KIT | Axitinib | 16.3642 | More.. |
| P10721 | KIT | Cabozantinib | 29.0162 | More.. |
| P10721 | KIT | Cediranib | 20.4673 | More.. |
| P10721 | KIT | Dasatinib | 16.1154 | More.. |
| P10721 | KIT | Imatinib | 21.287 | More.. |
| P10721 | KIT | Linifanib | 12.4093 | More.. |
| P10721 | KIT | Masitinib | 78.3859 | More.. |
| P10721 | KIT | Motesanib | 18.9152 | More.. |
| P10721 | KIT | OSI-930 | 83.3933 | More.. |
| P10721 | KIT | Pazopanib | 44.186 | More.. |
| P10721 | KIT | Sorafenib | 29.6257 | More.. |
| P10721 | KIT | Sunitinib | 34.8767 | More.. |
| P06239 | LCK | A-770041 | 22.6297 | More.. |
| P06239 | LCK | JW-7-24-1 | 18.1637 | More.. |
| P06239 | LCK | Staurosporine | 0.2727 | More.. |
| P06239 | LCK | WH-4-023 | 28.3974 | More.. |
| P53667 | LIMK1 | LIMK1 inhibitor BMS4 | 188.0383 | More.. |
| Q5S007 | LRRK2 | GSK2578215A | 237.1762 | More.. |
| P29376 | LTK | HG-5-113-01 | 8.989 | More.. |
| P29376 | LTK | XMD14-99 | 112.679 | More.. |
| O43318 | MAP3K7 | (5Z)-7-Oxozeaenol | 6.7243 | More.. |
| O43318 | MAP3K7 | NG-25 | 40.2513 | More.. |
| P41279 | MAP3K8 | KIN001-266 | 63.7041 | More.. |
| Q12851 | MAP4K2 | NG-25 | 40.2513 | More.. |
| Q13164 | MAPK7 | XMD8-92 | 40.4149 | More.. |
| P49137 | MAPKAPK2 | Staurosporine | 0.2727 | More.. |
| Q96L34 | MARK4 | XMD11-85h | 69.693 | More.. |
| P08581 | MET | AZD6094 | 26.9925 | More.. |
| P08581 | MET | Cabozantinib | 29.0162 | More.. |
| P08581 | MET | Crizotinib | 42.3076 | More.. |
| P08581 | MET | Foretinib | 7.1741 | More.. |
| P08581 | MET | JNJ38877605 | 106.7345 | More.. |
| P08581 | MET | PF2341066 | 6.5013 | More.. |
| P08581 | MET | PHA-665752 | 13.498 | More.. |
| P08581 | MET | Savolitinib | 23.9749 | More.. |
| P08581 | MET | SU11274 | 70.139 | More.. |
| Q9BUB5 | MKNK1 | ETP-45835 | 232.2917 | More.. |
| Q9HBH9 | MKNK2 | ETP-45835 | 232.2917 | More.. |
| Q04912 | MST1R | Foretinib | 7.1741 | More.. |
| P42345 | MTOR | JW-7-52-1 | 1.2292 | More.. |
| P42345 | MTOR | QL-VIII-58 | 1.1799 | More.. |
| P42345 | MTOR | Temsirolimus | 0.3619 | More.. |
| P42345 | MTOR | Voxtalisib | 111.0114 | More.. |
| P04629 | NTRK1 | AZD1332 | 60.7135 | More.. |
| P04629 | NTRK1 | GW441756 | 18.1112 | More.. |
| P04629 | NTRK1 | Lestaurtinib | 2.1852 | More.. |
| Q16620 | NTRK2 | AZD1332 | 60.7135 | More.. |
| Q16620 | NTRK2 | Lestaurtinib | 2.1852 | More.. |
| Q16620 | NTRK2 | WZ3105 | 6.3868 | More.. |
| Q16288 | NTRK3 | AZD1332 | 60.7135 | More.. |
| Q16288 | NTRK3 | Lestaurtinib | 2.1852 | More.. |
| O60285 | NUAK1 | WZ4003 | 122.9089 | More.. |
| Q9H093 | NUAK2 | WZ4003 | 122.9089 | More.. |
| Q13153 | PAK1 | IPA-3 | 167.2417 | More.. |
| Q13153 | PAK1 | PAK_5339 | 15.3624 | More.. |
| Q13177 | PAK2 | PAK_5339 | 15.3624 | More.. |
| P16234 | PDGFRA | Amuvatinib | 83.9825 | More.. |
| P16234 | PDGFRA | Masitinib | 78.3859 | More.. |
| P16234 | PDGFRA | Pazopanib | 44.186 | More.. |
| P16234 | PDGFRA | Ponatinib | 3.331 | More.. |
| P09619 | PDGFRB | Axitinib | 16.3642 | More.. |
| P09619 | PDGFRB | BIBF-1120 | 44.8965 | More.. |
| P09619 | PDGFRB | Brivanib, BMS-540215 | 117.5343 | More.. |
| P09619 | PDGFRB | Cediranib | 20.4673 | More.. |
| P09619 | PDGFRB | Dasatinib | 16.1154 | More.. |
| P09619 | PDGFRB | Foretinib | 7.1741 | More.. |
| P09619 | PDGFRB | Imatinib | 21.287 | More.. |
| P09619 | PDGFRB | Masitinib | 78.3859 | More.. |
| P09619 | PDGFRB | Motesanib | 18.9152 | More.. |
| P09619 | PDGFRB | Pazopanib | 44.186 | More.. |
| P09619 | PDGFRB | Sorafenib | 29.6257 | More.. |
| P09619 | PDGFRB | Sunitinib | 34.8767 | More.. |
| O15530 | PDPK1 | BX-912 | 41.945 | More.. |
| O15530 | PDPK1 | KIN001-244 | 57.4803 | More.. |
| O15530 | PDPK1 | OSU-03012 | 22.8051 | More.. |
| O15530 | PDPK1 | Staurosporine | 0.2727 | More.. |
| P42336 | PIK3CA | PI-103 | 26.7989 | More.. |
| P48736 | PIK3CG | Staurosporine | 0.2727 | More.. |
| P11309 | PIM1 | AZD1208 | 162.9102 | More.. |
| P11309 | PIM1 | SL0101 | 101.4104 | More.. |
| P11309 | PIM1 | Staurosporine | 0.2727 | More.. |
| Q9P1W9 | PIM2 | AZD1208 | 162.9102 | More.. |
| Q86V86 | PIM3 | AZD1208 | 162.9102 | More.. |
| Q86V86 | PIM3 | PI-103 | 26.7989 | More.. |
| Q86V86 | PIM3 | SL0101 | 101.4104 | More.. |
| P53350 | PLK1 | BI-2536 | 1.3712 | More.. |
| P53350 | PLK1 | GW843682X | 0.5363 | More.. |
| P53350 | PLK1 | MK-1775 | 6.0872 | More.. |
| P53350 | PLK1 | PLK_6522 | 0.5597 | More.. |
| Q9NYY3 | PLK2 | BI-2536 | 1.3712 | More.. |
| Q9NYY3 | PLK2 | PLK_6522 | 0.5597 | More.. |
| Q9H4B4 | PLK3 | BI-2536 | 1.3712 | More.. |
| Q9H4B4 | PLK3 | NPK76-II-72-1 | 52.3242 | More.. |
| Q9H4B4 | PLK3 | PLK_6522 | 0.5597 | More.. |
| P05771 | PRKCB | Enzastaurin | 74.1559 | More.. |
| Q05655 | PRKCD | XMD11-85h | 69.693 | More.. |
| Q04759 | PRKCQ | Staurosporine | 0.2727 | More.. |
| Q15139 | PRKD1 | kb NB 142-70 | 34.282 | More.. |
| P78527 | PRKDC | Voxtalisib | 111.0114 | More.. |
| P04049 | RAF1 | RAF_9304 | 19.6052 | More.. |
| P04049 | RAF1 | Sorafenib | 29.6257 | More.. |
| P07949 | RET | Cabozantinib | 29.0162 | More.. |
| P07949 | RET | Motesanib | 18.9152 | More.. |
| P07949 | RET | Sunitinib | 34.8767 | More.. |
| P07949 | RET | XMD11-85h | 69.693 | More.. |
| Q13546 | RIPK1 | XMD13-2 | 59.7873 | More.. |
| Q13464 | ROCK1 | GSK269962A | 17.6502 | More.. |
| Q13464 | ROCK1 | GSK429286A | 179.4792 | More.. |
| O75116 | ROCK2 | AZD5363 | 49.9909 | More.. |
| O75116 | ROCK2 | GSK269962A | 17.6502 | More.. |
| O75116 | ROCK2 | GSK429286A | 179.4792 | More.. |
| O75116 | ROCK2 | WZ3105 | 6.3868 | More.. |
| P08922 | ROS1 | Crizotinib | 42.3076 | More.. |
| P51812 | RPS6KA3 | CMK | 17.7762 | More.. |
| P51812 | RPS6KA3 | FMK | 193.3355 | More.. |
| P51812 | RPS6KA3 | SL0101 | 101.4104 | More.. |
| Q9HBY8 | SGK2 | GSK650394 | 81.3682 | More.. |
| Q96BR1 | SGK3 | GSK650394 | 81.3682 | More.. |
| P12931 | SRC | Bosutinib | 12.0191 | More.. |
| P12931 | SRC | Dasatinib | 16.1154 | More.. |
| P12931 | SRC | Ponatinib | 3.331 | More.. |
| P12931 | SRC | Saracatinib | 15.3916 | More.. |
| P12931 | SRC | WH-4-023 | 28.3974 | More.. |
| P12931 | SRC | WZ3105 | 6.3868 | More.. |
| Q96SB4 | SRPK1 | XMD11-85h | 69.693 | More.. |
| O94804 | STK10 | HG-5-113-01 | 8.989 | More.. |
| P43405 | SYK | BAY-61-3606 | 26.8765 | More.. |
| P43405 | SYK | Entospletinib | 86.6568 | More.. |
| P43405 | SYK | PRT062607 | 75.2024 | More.. |
| P43405 | SYK | Staurosporine | 0.2727 | More.. |
| P21675 | TAF1 | TAF1_5496 | 123.5989 | More.. |
| Q9UHD2 | TBK1 | BX795 | 15.6412 | More.. |
| P42680 | TEC | Bosutinib | 12.0191 | More.. |
| Q02763 | TEK | Cabozantinib | 29.0162 | More.. |
| Q02763 | TEK | Foretinib | 7.1741 | More.. |
| Q02763 | TEK | Ponatinib | 3.331 | More.. |
| P36897 | TGFBR1 | SB505124 | 87.8055 | More.. |
| P36897 | TGFBR1 | SB52334 | 123.3557 | More.. |
| P33981 | TTK | TTK_3146 | 23.9773 | More.. |
| O75385 | ULK1 | ULK1_4989 | 81.9118 | More.. |
| P30291 | WEE1 | MK-1775 | 6.0872 | More.. |
| P30291 | WEE1 | Wee1 Inhibitor | 29.3482 | More.. |
| P43403 | ZAP70 | Staurosporine | 0.2727 | More.. |